Compile Data Set for Download or QSAR
maximum 50k data
Found 52 of affinity data for UniProtKB/TrEMBL: Q1W675
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM22164((3R,5R)-7-[2-(4-fluorophenyl)-3-phenyl-4-(phenylca...)
Affinity DataIC50:  930nMAssay Description:Inhibition of pig liver microsomal HMG-CoA reductase by colorimetric methodMore data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50452901(CHEMBL4204041)
Affinity DataIC50:  5.82E+3nMAssay Description:Inhibition of pig liver microsomal HMG-CoA reductase by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50452895(CHEMBL4206214)
Affinity DataIC50:  6.21E+3nMAssay Description:Inhibition of pig liver microsomal HMG-CoA reductase by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50452899(CHEMBL4215012)
Affinity DataIC50:  6.76E+3nMAssay Description:Inhibition of pig liver microsomal HMG-CoA reductase by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50452894(CHEMBL4209384)
Affinity DataIC50:  7.43E+3nMAssay Description:Inhibition of pig liver microsomal HMG-CoA reductase by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50356919(CHEMBL1915760)
Affinity DataIC50:  8.60E+3nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50452891(CHEMBL4204038)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of pig liver microsomal HMG-CoA reductase by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50104745(Ganoderic acid DM)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50104745(Ganoderic acid DM)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50104764(CHEMBL3594152)
Affinity DataIC50:  1.07E+4nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50232011(CHEMBL4096720)
Affinity DataIC50:  1.23E+4nMAssay Description:Inhibition of pig liver microsomal HMG-CoA reductase by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50232011(CHEMBL4096720)
Affinity DataIC50:  1.23E+4nMAssay Description:Inhibition of HMG-CoA reductase in pig liver microsomes using HMG-CoA as substrate preincubated for 5 mins followed by NADPH addition measured after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50104746(Ganoderic Acid S)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50104766(CHEMBL3594158)
Affinity DataIC50:  1.26E+4nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50452892(CHEMBL4213527)
Affinity DataIC50:  1.32E+4nMAssay Description:Inhibition of pig liver microsomal HMG-CoA reductase by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50104765(CHEMBL3594153)
Affinity DataIC50:  1.33E+4nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50452898(CHEMBL4202495)
Affinity DataIC50:  1.42E+4nMAssay Description:Inhibition of pig liver microsomal HMG-CoA reductase by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50452889(CHEMBL4216288)
Affinity DataIC50:  1.65E+4nMAssay Description:Inhibition of pig liver microsomal HMG-CoA reductase by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50356923(CHEMBL1915763)
Affinity DataIC50:  1.68E+4nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50104754(CHEMBL3594142)
Affinity DataIC50:  1.71E+4nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50452896(CHEMBL4210421)
Affinity DataIC50:  1.81E+4nMAssay Description:Inhibition of pig liver microsomal HMG-CoA reductase by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50104748(CHEMBL3594154)
Affinity DataIC50:  1.89E+4nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50452897(CHEMBL4216284)
Affinity DataIC50:  1.89E+4nMAssay Description:Inhibition of pig liver microsomal HMG-CoA reductase by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50104759(CHEMBL3594147)
Affinity DataIC50:  2.05E+4nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50104749(CHEMBL3594155)
Affinity DataIC50:  2.41E+4nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50452893(CHEMBL4213110)
Affinity DataIC50:  2.51E+4nMAssay Description:Inhibition of pig liver microsomal HMG-CoA reductase by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50104763(CHEMBL3594151)
Affinity DataIC50:  2.64E+4nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50104756(CHEMBL3594144)
Affinity DataIC50:  2.66E+4nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50232007(GANOMYCIN B)
Affinity DataIC50:  2.93E+4nMAssay Description:Inhibition of HMG-CoA reductase in pig liver microsomes using HMG-CoA as substrate preincubated for 5 mins followed by NADPH addition measured after ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM22164((3R,5R)-7-[2-(4-fluorophenyl)-3-phenyl-4-(phenylca...)
Affinity DataIC50:  3.21E+4nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM22164((3R,5R)-7-[2-(4-fluorophenyl)-3-phenyl-4-(phenylca...)
Affinity DataIC50:  3.21E+4nMAssay Description:Inhibition of HMG-CoA reductase in pig liver microsomes using HMG-CoA as substrate preincubated for 5 mins followed by NADPH addition measured after ...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50104761(CHEMBL3594149)
Affinity DataIC50:  3.29E+4nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50452900(CHEMBL4216783)
Affinity DataIC50:  3.82E+4nMAssay Description:Inhibition of pig liver microsomal HMG-CoA reductase by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50232012(CHEMBL4067277)
Affinity DataIC50:  4.52E+4nMAssay Description:Inhibition of HMG-CoA reductase in pig liver microsomes using HMG-CoA as substrate preincubated for 5 mins followed by NADPH addition measured after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50452890(CHEMBL4211834)
Affinity DataIC50:  4.98E+4nMAssay Description:Inhibition of pig liver microsomal HMG-CoA reductase by colorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50232009(CHEMBL4094729)
Affinity DataIC50:  5.69E+4nMAssay Description:Inhibition of HMG-CoA reductase in pig liver microsomes using HMG-CoA as substrate preincubated for 5 mins followed by NADPH addition measured after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50104755(CHEMBL3594143)
Affinity DataIC50:  6.69E+4nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50104757(CHEMBL3594145)
Affinity DataIC50:  9.75E+4nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50232010(CHEMBL4087029)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HMG-CoA reductase in pig liver microsomes using HMG-CoA as substrate preincubated for 5 mins followed by NADPH addition measured after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50232008(fornicin C)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HMG-CoA reductase in pig liver microsomes using HMG-CoA as substrate preincubated for 5 mins followed by NADPH addition measured after ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50232006(CHEMBL4079168)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HMG-CoA reductase in pig liver microsomes using HMG-CoA as substrate preincubated for 5 mins followed by NADPH addition measured after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50232004(CHEMBL4104893)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HMG-CoA reductase in pig liver microsomes using HMG-CoA as substrate preincubated for 5 mins followed by NADPH addition measured after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50104768(CHEMBL3594159)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50104767(CHEBI:65945 | GANODERONE A)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50104751(CHEMBL3594157)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50104750(CHEMBL3594156)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50104762(CHEMBL3594150)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50104760(CHEMBL3594148)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50104758(CHEMBL3594146)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Sus scrofa)
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50104747(CHEMBL3594160)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of pig liver microsomes HMG-CoA reductase incubated for 5 mins in using HMG-CoA and NADPH by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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