BindingDB Data by Journal
PMID | Data | Article Title | Citation | Organization | Data Download |
---|---|---|---|---|---|
23327640 | 24 | Phenolic compounds with pancreatic lipase inhibitory activity from Korean yam (Dioscorea opposita).![]() | J Enzyme Inhib Med Chem 29: 1-6 (2014) | Seoul National University | 2D 3D TSV |
23323953 | 18 | Synthesis and carbonic anhydrase inhibitory properties of novel 1,4-dihydropyrimidinone substituted diarylureas.![]() | J Enzyme Inhib Med Chem 29: 18-22 (2014) | Sakarya University | 2D 3D TSV |
23311862 | 12 | Carbonic anhydrase inhibitory properties of novel sulfonamide derivatives of aminoindanes and aminotetralins.![]() | J Enzyme Inhib Med Chem 29: 35-42 (2014) | Atatürk University | 2D 3D TSV |
23323951 | 10 | Phenolic phytochemical displaying SARS-CoV papain-like protease inhibition from the seeds of Psoralea corylifolia.![]() | J Enzyme Inhib Med Chem 29: 59-63 (2014) | Gyeongsang National University | 2D 3D TSV |
23339426 | 46 | In vitro inhibition effect and structure-activity relationships of some saccharin derivatives on erythrocyte carbonic anhydrase I and II.![]() | J Enzyme Inhib Med Chem 29: 118-23 (2014) | Sakarya University | 2D 3D TSV |
23356363 | 215 | Benzenesulfonamides with benzimidazole moieties as inhibitors of carbonic anhydrases I, II, VII, XII and XIII.![]() | J Enzyme Inhib Med Chem 29: 124-31 (2014) | Vilnius University | 2D 3D TSV |
23356427 | 16 | Synthesis and carbonic anhydrase inhibitory properties of 1,3-dicarbonyl derivatives of methylaminobenzene-sulfonamide.![]() | J Enzyme Inhib Med Chem 29: 132-6 (2014) | Sakarya University | 2D 3D TSV |
23391138 | 14 | Synthesis and carbonic anhydrase isoenzymes I and II inhibitory effects of novel benzylamine derivatives.![]() | J Enzyme Inhib Med Chem 29: 168-74 (2014) | Atatürk University | 2D 3D TSV |
23534930 | 10 | Antileishmanial activity evaluation of bis-lawsone analogs and DNA topoisomerase-I inhibition studies.![]() | J Enzyme Inhib Med Chem 29: 185-9 (2014) | Karunya University | 2D 3D TSV |
23406473 | 4 | New chemotypes as Trypanosoma cruzi triosephosphate isomerase inhibitors: a deeper insight into the mechanism of inhibition.![]() | J Enzyme Inhib Med Chem 29: 198-204 (2014) | Universidad de la República | 2D 3D TSV |
23402383 | 6 | Discovery of new HER2/EGFR dual kinase inhibitors based on the anilinoquinazoline scaffold as potential anti-cancer agents.![]() | J Enzyme Inhib Med Chem 29: 215-22 (2014) | MSA University | 2D 3D TSV |
23432612 | 20 | Cytotoxicity and topoisomerase I/II inhibition activity of novel 4-aryl/alkyl-1-(piperidin-4-yl)-carbonylthiosemicarbazides and 4-benzoylthiosemicarbazides.![]() | J Enzyme Inhib Med Chem 29: 243-8 (2014) | Medical University | 2D 3D TSV |
23463940 | 4 | Synthesis and evaluation of 18F-labeled carbonic anhydrase IX inhibitors for imaging with positron emission tomography.![]() | J Enzyme Inhib Med Chem 29: 249-55 (2014) | BC Cancer Agency | 2D 3D TSV |
23488743 | 30 | Synthesis and dual D2 and 5-HT1A receptor binding affinities of 5-piperidinyl and 5-piperazinyl-1H-benzo[d]imidazol-2(3H)-ones.![]() | J Enzyme Inhib Med Chem 29: 281-91 (2014) | King Fahd University of Petroleum & Minerals | 2D 3D TSV |
23488741 | 20 | Novel coumarins and benzocoumarins acting as isoform-selective inhibitors against the tumor-associated carbonic anhydrase IX.![]() | J Enzyme Inhib Med Chem 29: 292-6 (2014) | S.G.S.I.T.S. | 2D 3D TSV |
23488740 | 12 | Novel inhibitor of bacterial sphingomyelinase, SMY-540, developed based on three-dimensional structure analysis.![]() | J Enzyme Inhib Med Chem 29: 303-10 (2014) | Tokushima Bunri University | 2D 3D TSV |
23578312 | 22 | Design, synthesis and evaluation of 2-phenylisothiazolidin-3-one-1,1-dioxides as a new class of human protein kinase CK2 inhibitors.![]() | J Enzyme Inhib Med Chem 29: 338-43 (2014) | NAS of Ukraine | 2D 3D TSV |
23663081 | 49 | Design, synthesis and biological evaluation of novel inosine 5'-monophosphate dehydrogenase (IMPDH) inhibitors.![]() | J Enzyme Inhib Med Chem 29: 408-19 (2014) | Nycomed | 2D 3D TSV |
23914927 | 24 | Inhibition of mammalian carbonic anhydrases I-XIV with grayanotoxin III: solution and in silico studies.![]() | J Enzyme Inhib Med Chem 29: 469-75 (2014) | University of Calgary | 2D 3D TSV |
23808805 | 42 | Carbonic anhydrase inhibitors. Phenols incorporating 2- or 3-pyridyl-ethenylcarbonyl and tertiary amine moieties strongly inhibit Saccharomyces cerevisiae ß-carbonic anhydrase.![]() | J Enzyme Inhib Med Chem 29: 495-9 (2014) | Ataturk University | 2D 3D TSV |
23895630 | 14 | Biochemical characterization of the chloroplastic ß-carbonic anhydrase from Flaveria bidentis (L.) "Kuntze".![]() | J Enzyme Inhib Med Chem 29: 500-4 (2014) | Istituto di Biostrutture e Bioimmagini-CNR | 2D 3D TSV |
24083411 | 7 | Effects of novel human cathepsin S inhibitors on cell migration in human cancer cells.![]() | J Enzyme Inhib Med Chem 29: 538-46 (2014) | National Tsing Hua University | 2D 3D TSV |
24090423 | 13 | Identification and structure-activity relationship study of carvacrol derivatives as Mycobacterium tuberculosis chorismate mutase inhibitors.![]() | J Enzyme Inhib Med Chem 29: 547-54 (2014) | Birla Institute of Technology | 2D 3D TSV |
25019596 | 24 | Quinolone-based HDAC inhibitors.![]() | J Enzyme Inhib Med Chem 29: 555-62 (2014) | Orchid Chemicals & Pharmaceuticals Limited | 2D 3D TSV |
24090419 | 36 | A systematic quantitative approach to rational drug design and discovery of novel human carbonic anhydrase IX inhibitors.![]() | J Enzyme Inhib Med Chem 29: 571-81 (2014) | Birla Institute of Technology | 2D 3D TSV |
24059701 | 21 | Discovery of a series of hydroximic acid derivatives as potent histone deacetylase inhibitors.![]() | J Enzyme Inhib Med Chem 29: 582-9 (2014) | Qingdao University | 2D 3D TSV |