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< Molecular Weight <
< KI (nM) <
< IC50 (nM) <
< ΔG° (kcal/mole) <
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0-9
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α-Carbonic anhydrase (αCA)
[
37
] [
3D
]
α-galactosidase
[
37
] [
3D
]
α-glucosidase
[
336
] [
3D
]
α7β2 nAChR
[
336
] [
3D
]
β-1,4-Galactosyltransferase I (β4GalT)
[
14
] [
3D
]
β-Carbonic anhydrase (βCA)
[
14
] [
3D
]
β-Carbonic anhydrase (CA)
[
14
] [
3D
]
β-Carbonic anhydrase (CA1)
[
14
] [
3D
]
β-Carbonic anhydrase 2 (CA 2)
[
62
] [
3D
]
β-Carbonic anhydrase 3 (CA 3)
[
62
] [
3D
]
β-galactosidase
[
101
] [
3D
]
β-glucosidase
[
101
] [
3D
]
β-ketoacyl-ACP synthase I (C171Q KasA)
[
1
] [
3D
]
β-Ketoacyl-acyl carrier protein (ACP) synthase III (FabH)
[
1
] [
3D
]
β-lactamase (Bla2)
[
20
] [
3D
]
κ opioid receptor (KOR D138A)
[
20
] [
3D
]
κ opioid receptor (KOR D138N)
[
5
] [
3D
]
κ opioid receptor (KOR E297A)
[
5
] [
3D
]
κ opioid receptor (KOR H291A)
[
5
] [
3D
]
κ opioid receptor (KOR H291F)
[
5
] [
3D
]
κ opioid receptor (KOR I135A)
[
5
] [
3D
]
κ opioid receptor (KOR I294A)
[
5
] [
3D
]
κ opioid receptor (KOR I316A)
[
5
] [
3D
]
κ opioid receptor (KOR K200A)
[
5
] [
3D
]
κ opioid receptor (KOR K227A)
[
5
] [
3D
]
κ opioid receptor (KOR L212A)
[
5
] [
3D
]
κ opioid receptor (KOR M142A)
[
5
] [
3D
]
κ opioid receptor (KOR M226A)
[
5
] [
3D
]
κ opioid receptor (KOR Q115A)
[
5
] [
3D
]
κ opioid receptor (KOR Y119A)
[
5
] [
3D
]
κ opioid receptor (KOR Y119F)
[
5
] [
3D
]
κ opioid receptor (KOR Y139A)
[
5
] [
3D
]
κ opioid receptor (KOR Y139F)
[
5
] [
3D
]
κ opioid receptor (KOR Y312A)
[
5
] [
3D
]
κ opioid receptor (KOR Y312F)
[
5
] [
3D
]
κ opioid receptor (KOR Y313A)
[
5
] [
3D
]
κ opioid receptor (KOR Y313F)
[
5
] [
3D
]
κ opioid receptor (KOR Y320A)
[
5
] [
3D
]
κ opioid receptor (KOR Y320F)
[
5
] [
3D
]
κ opioid receptor (KOR Y66A)
[
5
] [
3D
]
σB-DNA
[
1
] [
3D
]
α-Amylase group 4 allergen (Aca s 4)
[
1
] [
3D
]
(E)-1-hydroxy-2-methyl-but-2-enyl 4-diphosphate reductase (IspH)
[
2
] [
3D
]
1,3-beta-glucan synthase
[
2
] [
3D
]
1,3-beta-glucan synthase component GLS2
[
988
] [
3D
]
1,4-Dihydroxy-2-naphthoyl-CoA synthase
[
988
] [
3D
]
1,5-anhydro-D-fructose reductase
[
69
] [
3D
]
1-acylglycerol-3-phosphate O-acyltransferase beta
[
69
] [
3D
]
1-deoxy-D-xylulose 5-phosphate reductoisomerase
[
183
] [
3D
]
1-deoxy-D-xylulose-5-phosphate synthase
[
183
] [
3D
]
1-Deoxy-D-xylulose-5-phosphate synthase (DXP synthase))
[
8
] [
3D
]
1-deoxyxylulose-5-phosphate reductoisomerase
[
8
] [
3D
]
1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase delta-1
[
3
] [
3D
]
1-phosphatidylinositol-4,5-bisphosphate phosphodiesterase gamma-1
[
3
] [
3D
]
11-beta-hydroxysteroid dehydrogenase 1
[
3379
] [
3D
]
11-beta-Hydroxysteroid Dehydrogenase 1 (11-beta-HSD1)
[
1
] [
3D
]
11-beta-hydroxysteroid dehydrogenase 2
[
494
] [
3D
]
11-beta-Hydroxysteroid Dehydrogenase 2 (11-beta-HSD2)
[
494
] [
3D
]
11-beta-hydroxysteroid dehydrogenase type 1
[
2
] [
3D
]
12-Lipoxygenase (12-LOX)
[
2
] [
3D
]
14-3-3 protein beta/alpha
[
1
] [
3D
]
14-3-3 protein eta
[
1
] [
3D
]
14-3-3 protein sigma
[
2
] [
3D
]
14-3-3 protein theta
[
2
] [
3D
]
14-3-3 protein zeta/delta
[
17
] [
3D
]
14-alpha sterol demethylase
[
17
] [
3D
]
14-alpha sterol demethylase Cyp51A
[
5
] [
3D
]
15-hydroxyprostaglandin dehydrogenase [NAD(+)]
[
5
] [
3D
]
15-hydroxyprostaglandin dehydrogenase [NAD+]
[
366
] [
3D
]
15-Lipoxygenase (LoxA)
[
366
] [
3D
]
15-Lipoxygenase (SLO)
[
13
] [
3D
]
15-Lipoxygenase-2 (15-LOX-2)
[
13
] [
3D
]
17-beta-Hydroxysteroid Dehydrogenase 1 (17-beta-HSD1)
[
44
] [
3D
]
17-beta-hydroxysteroid dehydrogenase 14
[
44
] [
3D
]
17-beta-Hydroxysteroid Dehydrogenase 5 (17-beta-HSD5, AKR1C3)
[
492
] [
3D
]
17-beta-hydroxysteroid dehydrogenase type 3
[
492
] [
3D
]
17-beta-hydroxysteroid-dehydrogenase
[
12
] [
3D
]
2'-deoxynucleoside 5'-phosphate N-hydrolase 1
[
12
] [
3D
]
2,3-dihydroxybenzoate-AMP ligase
[
102
] [
3D
]
2,6-dichloro-p-hydroquinone 1,2-dioxygenase (PcpA)
[
102
] [
3D
]
2-acylglycerol O-acyltransferase 2
[
2
] [
3D
]
2-amino-3-carboxymuconate-6-semialdehyde decarboxylase
[
2
] [
3D
]
2-amino-4-hydroxy-6-hydroxymethyldihydropteridin e pyrophosphokinase
[
60
] [
3D
]
2-amino-4-hydroxy-6-hydroxymethyldihydropteridine pyrophosphokinase
[
60
] [
3D
]
2-C-methyl-D-erythritol 2,4-cyclodiphosphate synthase
[
7
] [
3D
]
2-dehydro-3-deoxyphosphooctonate aldolase
[
7
] [
3D
]
2-heptyl-4(1H)-quinolone synthase PqsD
[
34
] [
3D
]
2-oxoglutarate receptor 1
[
34
] [
3D
]
20-alpha-Hydroxysteroid Dehydrogenase (AKR1C1) Mutant (H222S)
[
1
] [
3D
]
20-alpha-Hydroxysteroid Dehydrogenase (AKR1C1) Mutant (L306A)
[
1
] [
3D
]
20-alpha-Hydroxysteroid Dehydrogenase (AKR1C1) Mutant (L308A)
[
1
] [
3D
]
20-alpha-Hydroxysteroid Dehydrogenase (AKR1C1) Mutant (L54V)
[
1
] [
3D
]
20S proteasome
[
2
] [
3D
]
20S proteasome chymotrypsin-like
[
2
] [
3D
]
24-sterol C-methyltransferase
[
49
] [
3D
]
25-hydroxyvitamin D-1 alpha hydroxylase, mitochondrial
[
49
] [
3D
]
26S Proteasome regulatory subunit Rpn11 (Rpn11)
[
478
] [
3D
]
26S proteosome
[
478
] [
3D
]
2C-methyl-D-erythritol-2,4-cyclodiphosphate synthase (IspF)
[
9
] [
3D
]
3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase
[
9
] [
3D
]
3',5'-cyclic phosphodiesterase
[
663
] [
3D
]
3',5'-cyclic phosphodiesterase (PDE2A)
[
663
] [
3D
]
3-beta-hydroxysteroid dehydrogenase/delta 5-->4-isomerase type I
[
15
] [
3D
]
3-beta-hydroxysteroid dehydrogenase/delta 5-->4-isomerase type II
[
15
] [
3D
]
3-beta-hydroxysteroid-delta(8),delta(7)-isomerase
[
115
] [
3D
]
3-dehydroquinate dehydratase
[
115
] [
3D
]
3-dehydroquinate synthase
[
10
] [
3D
]
3-deoxy-D-arabino-heptulosonate 7-phosphate synthase, Phe-sensitive
[
10
] [
3D
]
3-hydroxy-3-methylglutaryl-coenzyme A reductase
[
72
] [
3D
]
3-hydroxy-3-methylglutaryl-coenzyme A reductase (HMG-CoA)
[
72
] [
3D
]
3-hydroxyanthranilate 3,4-dioxygenase
[
1
] [
3D
]
3-Hydroxybenzoate 6-hydroxylase (3HB6H H213A)
[
1
] [
3D
]
3-Hydroxybenzoate 6-hydroxylase (3HB6H Y105F)
[
1
] [
3D
]
3-Hydroxybenzoate 6-hydroxylase (3HB6H)
[
1
] [
3D
]
3-keto-steroid reductase
[
3
] [
3D
]
3-oxoacyl-(Acyl-carrier protein) reductase
[
3
] [
3D
]
3-oxoacyl-acyl-carrier protein reductase
[
15
] [
3D
]
3-oxoacyl-[acyl-carrier-protein] synthase 1
[
15
] [
3D
]
3-oxoacyl-[acyl-carrier-protein] synthase 2
[
38
] [
3D
]
3-phosphoinositide dependent protein kinase-1
[
38
] [
3D
]
3-phosphoinositide-dependent protein kinase 1 (51-359)
[
781
] [
3D
]
3-Phosphoinositide-Dependent Protein Kinase 1 (PDK1)
[
781
] [
3D
]
3-Phosphoinositide-Dependent Protein Kinase 1 (PDK1) Mutant (A162V)
[
2
] [
3D
]
3-Phosphoinositide-Dependent Protein Kinase 1 (PDK1) Mutant (E166D)
[
2
] [
3D
]
3-Phosphoinositide-Dependent Protein Kinase 1 (PDK1) Mutant (L159M)
[
2
] [
3D
]
3-Phosphoinositide-Dependent Protein Kinase 1 (PDK1) Mutant (T222A)
[
2
] [
3D
]
3-Phosphoinositide-Dependent Protein Kinase 1 (PDK1) Mutant (V143T)
[
2
] [
3D
]
3-Phosphoinositide-Dependent Protein Kinase 1 (PDK1) Mutant (V143T/T222A)
[
2
] [
3D
]
3C-like protease
[
101
] [
3D
]
3C-like proteinase (3CL-PRO)
[
101
] [
3D
]
3C-like proteinase (CVB3 3Cpro)
[
5
] [
3D
]
4,4'-diapophytoene desaturase (4,4'-diaponeurosporene-forming)
[
5
] [
3D
]
4-diphosphocytidyl-2-C-methyl-D-erythritol kinase
[
6
] [
3D
]
4-hydroxy-2-oxoglutarate aldolase, mitochondrial
[
6
] [
3D
]
4-hydroxyphenylpyruvate dioxygenase
[
161
] [
3D
]
40S ribosomal protein S27
[
161
] [
3D
]
5'-AMP-activated protein kinase subunit beta-1
[
20
] [
3D
]
5'-AMP-activated protein kinase subunit gamma-1
[
20
] [
3D
]
5α-Reductase 1 (5α-R1)
[
433
] [
3D
]
5' exonuclease Apollo
[
433
] [
3D
]
5'-AMP-activated protein kinase catalytic subunit alpha-1
[
125
] [
3D
]
5'-AMP-activated protein kinase catalytic subunit alpha-1/beta-1/gamma-1
[
125
] [
3D
]
5'-AMP-activated protein kinase catalytic subunit alpha-2/beta-1/gamma-2
[
2
] [
3D
]
5'-AMP-activated protein kinase Complex 1
[
2
] [
3D
]
5'-AMP-activated protein kinase subunit gamma-2
[
1
] [
3D
]
5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase
[
1
] [
3D
]
5-alpha-Reductase (5α-Reductase)
[
12
] [
3D
]
5-enolpyruvylshikimate-3-phosphate synthase
[
12
] [
3D
]
5-HT1
[
21
] [
3D
]
5-HT1 like
[
21
] [
3D
]
5-HT1A/ 5-HT2c
[
5
] [
3D
]
5-HT2
[
5
] [
3D
]
5-HT3A Serotonin Receptor
[
169
] [
3D
]
5-HT5
[
169
] [
3D
]
5-HT5B
[
29
] [
3D
]
5-hydroxytryptamine 1D receptor (5HT1D)
[
29
] [
3D
]
5-hydroxytryptamine receptor 1A (5-HT1A)
[
4674
] [
3D
]
5-hydroxytryptamine receptor 1A (5HT1A)
[
1
] [
3D
]
5-hydroxytryptamine receptor 1A (5HT1B)
[
1
] [
3D
]
5-hydroxytryptamine receptor 1B
[
1
] [
3D
]
5-hydroxytryptamine receptor 1B (5HT1B)
[
61
] [
3D
]
5-hydroxytryptamine receptor 1D
[
61
] [
3D
]
5-hydroxytryptamine receptor 1D (5HT1D)
[
6
] [
3D
]
5-hydroxytryptamine receptor 2A
[
6
] [
3D
]
5-hydroxytryptamine receptor 2A (5HT2A)
[
72
] [
3D
]
5-hydroxytryptamine receptor 2B
[
72
] [
3D
]
5-hydroxytryptamine receptor 2B (5HT2B)
[
32
] [
3D
]
5-hydroxytryptamine receptor 2C
[
32
] [
3D
]
5-hydroxytryptamine receptor 2C (5HT2C)
[
13
] [
3D
]
5-hydroxytryptamine receptor 3A
[
13
] [
3D
]
5-hydroxytryptamine receptor 4 (5-HT4)
[
401
] [
3D
]
5-hydroxytryptamine receptor 4 (5-HT4e)
[
401
] [
3D
]
5-Hydroxytryptamine receptor 6 (5-HT6)
[
3025
] [
3D
]
5-Hydroxytryptamine receptor 7 (5-HT7)
[
1
] [
3D
]
5-hydroxytryptamine receptor 7 (5HT7)
[
29
] [
3D
]
5-Lipoxygenase
[
29
] [
3D
]
5-Lipoxygenase (5-LOX)
[
5
] [
3D
]
5-lipoxygenase-activating protein (FLAP)
[
5
] [
3D
]
5-Lipoxygenase/5-lipoxygenase activating protein
[
20
] [
3D
]
5-lipoxygenase/FLAP
[
20
] [
3D
]
6,7-dimethyl-8-ribityllumazine synthase
[
8
] [
3D
]
6-O-methylguanine-DNA methyltransferase
[
8
] [
3D
]
6-phospho-1-fructokinase
[
53
] [
3D
]
6-phospho-1-fructokinase, putative
[
53
] [
3D
]
6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 1
[
37
] [
3D
]
6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 2
[
37
] [
3D
]
6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 3 (PFKFB3)
[
106
] [
3D
]
6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 4 (PFKFB4)
[
106
] [
3D
]
6-phosphogluconate dehydrogenase (6PGD)
[
29
] [
3D
]
6-phosphogluconate dehydrogenase, decarboxylating
[
29
] [
3D
]
6-phosphogluconate dehydrogenase, decarboxylating, putative
[
5
] [
3D
]
6-phosphogluconolactonase
[
5
] [
3D
]
60 kDa heat shock protein, mitochondrial
[
2
] [
3D
]
7-dehydrocholesterol reductase
[
2
] [
3D
]
72 kDa type IV collagenase
[
4448
] [
3D
]
78 kDa glucose-regulated protein
[
1
] [
3D
]
8-Oxoguanine DNA glycosylase-1 (OGG1)
[
20
] [
3D
]