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Targets Binding with 108 Compounds
Target Name
Affinity Link(s)
Article(s)
UniProt
Files
Cysteinyl leukotriene receptor 2
Ki:
8
IC50:
115
8
4
2D
3D
TSV
Glutathione S-transferase P/Tyrosine-protein kinase JAK1
IC50:
111
1
7
2D
3D
TSV
Glutathione S-transferase P/Tyrosine-protein kinase JAK2
IC50:
111
1
7
2D
3D
TSV
GTPase KRas [G12C]
IC50:
126
2
6
2D
3D
TSV
Histone deacetylase 1/2/3/8
IC50:
77
EC50:
74
14
25
2D
3D
TSV
Leukotriene C4 synthase
IC50:
200
7
5
2D
3D
TSV
Proto-oncogene tyrosine-protein kinase receptor Ret [658-1114,G810R]
IC50:
110
1
7
2D
3D
TSV
Putative P2Y purinoceptor 10
EC50:
202
3
8
2D
3D
TSV
Pyruvate kinase
IC50:
109
5
2
2D
3D
TSV
Salicyl-AMP ligase / salicyl-S-ArCP synthetase
Ki:
110
IC50:
1
Kd:
1
7
5
2D
3D
TSV
Similar to alpha-tubulin isoform 1/Tubulin beta-2B chain
IC50:
108
EC50:
6
8
3
2D
3D
TSV
Tryptophan 5-hydroxylase 2
IC50:
144
EC50:
4
6
5
2D
3D
TSV