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Targets Binding with 40 Compounds
Target Name
Affinity Link(s)
Article(s)
UniProt
Files
3-oxoacyl-ACP synthase
IC50:
41
Kd:
1
4
3
2D
3D
TSV
Arginase
Ki:
17
IC50:
32
Kd:
7
6
3
2D
3D
TSV
Bacterial leucyl aminopeptidase
Ki:
25
IC50:
17
5
1
2D
3D
TSV
Beta-arrestin-1
Ki:
37
IC50:
1
EC50:
11
9
9
2D
3D
TSV
Casein kinase II subunit alpha'/beta
Ki:
4
IC50:
37
2
6
2D
3D
TSV
Cathepsin L
Ki:
40
2
2
2D
3D
TSV
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A [388-1112]
IC50:
40
1
5
2D
3D
TSV
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3B [387-1112]
IC50:
40
1
6
2D
3D
TSV
Chitinase B
Ki:
4
IC50:
44
Kd:
2
9
1
2D
3D
TSV
Cyclin-dependent kinase/G1/S-specific cyclin- 2
IC50:
76
2
9
2D
3D
TSV
Cystine/glutamate transporter
Ki:
7
IC50:
47
5
3
2D
3D
TSV
Delta carbonic anhydrase
Ki:
40
1
1
2D
3D
TSV
Delta-aminolevulinic acid dehydratase
Ki:
21
IC50:
54
EC50:
12
4
16
2D
3D
TSV
E3 ubiquitin-protein ligase XIAP [1-168]/[124-242]
Ki:
48
1
6
2D
3D
TSV
Egl nine homolog 1 [179-426]
IC50:
41
2
5
2D
3D
TSV
Epidermal growth factor receptor [1-18,20-1210,T790M]
IC50:
40
2
17
2D
3D
TSV
Epidermal growth factor receptor [1-18,20-1210]
IC50:
40
2
16
2D
3D
TSV
Epidermal growth factor receptor/Receptor tyrosine-protein kinase erbB-2
IC50:
40
3
21
2D
3D
TSV
Glutaminase liver isoform, mitochondrial
IC50:
40
5
9
2D
3D
TSV
Glutathione hydrolase 1 proenzyme
Ki:
7
IC50:
33
4
10
2D
3D
TSV
Integrin alpha-4/Integrin beta-1/Vascular cell adhesion protein 1
IC50:
40
1
25
2D
3D
TSV
MAP kinase-activated protein kinase 3
Ki:
2
IC50:
39
24
3
2D
3D
TSV
Probable C-C chemokine receptor type 3
Ki:
32
IC50:
12
7
3
2D
3D
TSV
Probable G-protein coupled receptor 174
EC50:
67
1
3
2D
3D
TSV
Protein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type
IC50:
41
4
15
2D
3D
TSV
Protein mono-ADP-ribosyltransferase PARP6
IC50:
40
6
7
2D
3D
TSV
Sodium/potassium-transporting ATPase subunit alpha-1/beta-1
Ki:
44
IC50:
4
4
16
2D
3D
TSV
Sodium/potassium-transporting ATPase subunit alpha-2/beta-1
Ki:
44
IC50:
4
4
11
2D
3D
TSV
Sphingomyelin phosphodiesterase 2
Ki:
2
IC50:
47
6
6
2D
3D
TSV
Tyrosine-protein kinase SYK [2-635]
IC50:
40
3
1
2D
3D
TSV