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PMIDDataArticle TitleCitationOrganizationSD Files Download
995128 168 Properties of [3H]haloperidol and [3H]dopamine binding associated with dopamine receptors in calf brain membranes.BDB Mol Pharmacol 12: 800-12 (1976) TBA 2D 3D TSV
950651 6 Synthesis and properties of 2-S-(N,N-dialkylamino)ethyl)thio-1,3,2-dioxaphosphorinane 2-oxide and of the corresponding quaternary derivatives as potential nontoxic antiglaucoma agents.EBI J Med Chem 19: 810-3 (1976) TBA 2D 3D TSV
926113 5 Synthesis and biological action of two glucocorticoid alkylating agents.EBI J Med Chem 20: 1134-9 (1978) TBA 2D 3D TSV
915907 6 Proteinase inhibitors. I. Inhibitors of elastase.EBI J Med Chem 20: 1464-8 (1977) TBA 2D 3D TSV
903914 7 Synthesis and evaluation of alpha-hydroxythiol esters as antitumor agents and glyoxalase I inhibitors.EBI J Med Chem 20: 1239-42 (1977) TBA 2D 3D TSV
874952 1 New inhibitors of steroid 11beta-hydroxylase. Structure--activity relationship studies of metyrapone-like compounds.EBI J Med Chem 20: 762-6 (1977) TBA 2D 3D TSV
850237 38 Synthesis and structure-activity relationships of bestatin analogues, inhibitors of aminopeptidase B.EBI J Med Chem 20: 510-5 (1977) TBA 2D 3D TSV
850236 1 Inhibition of histidine decarboxylase. Derivatives of histidine.EBI J Med Chem 20: 506-9 (1977) TBA 2D 3D TSV
782880 21 Influence of side-chain structure of aliphatic amino acids on binding to isoleucyl-tRNA synthetase from Escherichia coli MRE 600.BDB Eur J Biochem 66: 147-55 (1976) Gesellschaft Fur Molekularbiolische Forschung mbH 2D 3D TSV
722762 2 Effects of thiophene analogues of chloroamphetamines on central serotonergic mechanisms.EBI J Med Chem 21: 978-81 (1979) TBA 2D 3D TSV
722731 1 Prodrugs of 9-beta-D-arabinofuranosyladenine. 1. Synthesis and evaluation of some 5'-(O-acyl) derivatives.EBI J Med Chem 21: 1218-21 (1979) TBA 2D 3D TSV
722719 1 Use of adenine nucleotide derivatives to assess the potential of exo-active-site-directed reagents as species- or isozyme-specific enzyme inactivators. 2. Isozyme-specific inactivation of a mammalian enzyme and its significance in the possible design of fetal isozyme targeted antineoplastic agents.EBI J Med Chem 21: 1137-40 (1979) TBA 2D 3D TSV
722718 56 Structure-activity relationships for the inhibition of acrosin by benzamidine derivatives.EBI J Med Chem 21: 1132-6 (1979) TBA 2D 3D TSV
722711 5 Synthesis and biochemical evaluation of inhibitors of estrogen biosynthesis.EBI J Med Chem 21: 1007-11 (1979) TBA 2D 3D TSV
671460 122 Diarylamidine derivatives with one or both of the aryl moieties consisting of an indole or indole-like ring. Inhibitors of arginine-specific esteroproteases.EBI J Med Chem 21: 613-23 (1978) TBA 2D 3D TSV
660589 3 Inactivation of trypsin-like proteases by sulfonylation. Variation of positively charged group and inhibitor length.EBI J Med Chem 21: 456-9 (1978) TBA 2D 3D TSV
619149 20 Analogues of ornithine as inhibitors of ornithine decarboxylase. New deductions concerning the topography of the enzyme's active site.EBI J Med Chem 21: 50-5 (1978) TBA 2D 3D TSV
592342 45 Hypolipidemic activity of 5-aryl-3-methylvaleric acid derivatives.EBI J Med Chem 20: 1705-8 (1978) TBA 2D 3D TSV
592327 104 Potent reversible anticholinesterase agents. Bis- and mono-N-substituted benzoquinolinium halides.EBI J Med Chem 20: 1617-23 (1978) TBA 2D 3D TSV
559765 2 Vitamin B6 antagonists obtained by replacing or modifying the 2-methyl group.EBI J Med Chem 20: 745-9 (1977) TBA 2D 3D TSV
557561 3 4-Halovinyl- and 4-ethynyl-4-deformylpyridoxal derivatives and related analogues as potentially irreversible antagonists of vitamin B6.EBI J Med Chem 20: 567-72 (1977) TBA 2D 3D TSV
556774 58 Inhibition of acetylcholinesterase by thiamine. A structure-function study.EBI J Med Chem 20: 161-4 (1977) TBA 2D 3D TSV
556772 1 Antagonists of vitamin B6. Simultaneous and stepwise modification of the 2 and 4 positions.EBI J Med Chem 20: 1-5 (1977) TBA 2D 3D TSV
533888 1 Synthesis and biological evaluation of 9,11-azo-13-oxa-15-hydroxyprostanoic acid, a potent inhibitor of platelet aggregation.EBI J Med Chem 22: 1402-8 (1980) TBA 2D 3D TSV
533882 1 Synthesis of spiro[isobenzofuran-1(3H),4'-piperidines] as potential central nervous system agents. 5. Conformationally mobile analogues derived by furan ring opening.EBI J Med Chem 22: 1347-54 (1980) TBA 2D 3D TSV
490541 1 Synthesis and antiestrogenic activity of [3,4-dihydro-2-(4-methoxyphenyl)-1-naphthalenyl][4-[2-(1-pyrrolidinyl)ethoxy]-phenyl]methanone, methanesulfonic acid salt.EBI J Med Chem 22: 962-6 (1979) TBA 2D 3D TSV
459687 7 Evidence for two types of binding of 3H-gaba and 3H-muscimol in rat cerebral cortex and cerebellum.BDB Life Sci 24: 1849-54 (1979) TBA 2D 3D TSV
458818 26 Design of species- or isozyme-specific enzyme inhibitors. 1. Effect of thymidine substituents on affinity for the thymidine site of hamster cytoplasmic thymidine kinase.EBI J Med Chem 22: 621-31 (1979) TBA 2D 3D TSV
430474 2 trans-5-(3,3,3-Trifluoro-1-propenyl-)-2'-deoxyuridylate: a mechanism-based inhibitor of thymidylate synthetase.EBI J Med Chem 22: 339-40 (1979) TBA 2D 3D TSV
430054 14 Characterization of the binding of [3H]muscimol, a potent gamma-aminobutyric acid agonist, to rat brain synaptosomal membranes using a filtration assay.BDB J Neurochem 32: 713-8 (1979) TBA 2D 3D TSV
423213 22 Inhibition of gastric acid secretion by 1,8-naphthyridin-2(1H)-ones.EBI J Med Chem 22: 301-6 (1979) TBA 2D 3D TSV
423205 119 Cyclic amidine inhibitors of indolamine N-methyltransferase.EBI J Med Chem 22: 237-47 (1979) TBA 2D 3D TSV
423204 2 Coenzyme--substrate adducts as inhibitors of mouse liver 3,4-dihydroxyphenylalanine decarboxylase.EBI J Med Chem 22: 233-7 (1979) TBA 2D 3D TSV
423172 1 Phosphonate analogue of 2'-deoxy-5-fluorouridylic acid.EBI J Med Chem 22: 109-11 (1979) TBA 2D 3D TSV
410930 15 Inhibition of Lactobacillus casei thymidylate synthetase by 5-substituted 2'-deoxyuridylates. Preliminary quantitative structure-activity relationship.EBI J Med Chem 20: 1469-73 (1977) TBA 2D 3D TSV
409842 24 Methotrexate analogues. 9. Synthesis and biological properties of some 8-alkyl-7,8-dihydro analogues.EBI J Med Chem 20: 1323-7 (1977) TBA 2D 3D TSV
323484 8 Thymidylate synthetase inhibitors. Synthesis of N-substituted 5-aminomethyl-2'-deoxyuridine 5'-phosphates.EBI J Med Chem 20: 669-73 (1977) TBA 2D 3D TSV
321782 9 A manual method for applying the Hansch approach to drug design.EBI J Med Chem 20: 463-9 (1977) TBA 2D 3D TSV
282646 50 Histamine H1 receptors identified in mammalian brain membranes with [3H]mepyramine.BDB Proc Natl Acad Sci U S A 75: 6290-4 (1978) TBA 2D 3D TSV
231655 18 Design of species- or isozyme-specific enzyme inhibitors. 3. Species and isozymic differences between mammalian and bacterial adenylate kinases in substituent tolerance in an enzyme-substrate complex.EBI J Med Chem 22: 1529-32 (1980) TBA 2D 3D TSV
226705 4 Synthesis and biological properties of N2-substituted spin-labeled analogues of actinomycin D.EBI J Med Chem 22: 1051-5 (1979) TBA 2D 3D TSV
199727 8 Synthesis of beta-spiro[pyrrolidinoindolines], their binding to the glycine receptor, and in vivo biological acitivity.EBI J Med Chem 20: 1448-51 (1977) TBA 2D 3D TSV
184284 1 Synthesis and biological properties of some spin-labeled 9-aminoacridines.EBI J Med Chem 19: 994-8 (1976) TBA 2D 3D TSV
152812 69 Inhibition of four human serine proteases by substituted benzamidines.EBI J Med Chem 21: 1202-7 (1979) TBA 2D 3D TSV
114660 8 5-Cyano-2'-deoxyuridine 5'-phosphate: a potent competitive inhibitor of thymidylate synthetase.EBI J Med Chem 22: 1137-9 (1979) TBA 2D 3D TSV
110934 12 Synthesis and biological activity of 8-oxadihydropteridines.EBI J Med Chem 22: 741-3 (1979) TBA 2D 3D TSV
110931 2 Synthesis of 5-selenium-substituted uracil derivatives. Inhibition of thymidylate synthetase by 5-hydroseleno-2'-deoxyuridylate.EBI J Med Chem 22: 618-21 (1979) TBA 2D 3D TSV
109616 9 Methotrexate analogues. 12. Synthesis and biological properties of some aza homologues.EBI J Med Chem 22: 869-74 (1979) TBA 2D 3D TSV
106122 3 Enzyme affinity of the 5,6-dihydro derivatives of the substrate and product of thymidylate synthetase catalysis.EBI J Med Chem 22: 319-21 (1979) TBA 2D 3D TSV
40029 1 Absolute configuration of glycerol derivatives. 7. Enantiomers of 2-[[[2-(2,6-dimethoxyphenoxy)ethyl]amino]methyl]-1,4-benzodioxane (WB-4101), a potent competitive alpha-adrenergic antagonist.EBI J Med Chem 22: 1125-7 (1979) TBA 2D 3D TSV
40025 4 Nicotinamide adenine dinucleotide phosphate-decanaldehyde adduct as an inhibitor of beef brain NADP-linked aldehyde reductase.EBI J Med Chem 22: 1011-4 (1979) TBA 2D 3D TSV
37098 14 Binding characteristics of 3H-prazosin to rat brain alpha-adrenergic receptors.BDB Eur J Pharmacol 55: 323-6 (1979) TBA 2D 3D TSV
31484 4 Stereoelectronic factors in the binding of substrate analogues and inhibitors to purine nucleoside phosphorylase isolated from human erythrocytes.EBI J Med Chem 21: 877-82 (1979) TBA 2D 3D TSV
22757 12 Antidepressant agents. 9. 3,3-Diphenylcyclobutylamines, a new class of central stimulants.EBI J Med Chem 21: 78-82 (1978) TBA 2D 3D TSV
20632 7 Specific benzodiazepine receptors in rat brain characterized by high-affinity (3H)diazepam binding.BDB Proc Natl Acad Sci U S A 74: 3805-9 (1977) TBA 2D 3D TSV
17827 156 Binding characteristics of a radiolabeled agonist and antagonist at central nervous system alpha noradrenergic receptors.BDB Mol Pharmacol 13: 454-73 (1977) TBA 2D 3D TSV
8699 51 Beta adrenergic receptor binding in membrane preparations from mammalian brain.BDB Mol Pharmacol 12: 568-80 (1976) TBA 2D 3D TSV
7724 61 Alpha-noradrenergic receptor binding in mammalian brain: differential labeling of agonist and antagonist states.BDB Life Sci 19: 69-76 (1976) TBA 2D 3D TSV
2778 28 Synthesis and enzymic activity of some novel xanthine oxidase inhibitors. 3-Substituted 5,7-dihydroxypyrazolo(1,5-alpha)pyrimidines.EBI J Med Chem 19: 291-6 (1976) TBA 2D 3D TSV
1535 2 Conformationally restricted analogs of histamine H1 receptor antagonists: trans and cis-1-benzyl-3-dimethylamino-6-phenylpiperidine.EBI J Med Chem 19: 117-22 (1976) TBA 2D 3D TSV

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