PMID

Data

Article Title

Organization

Synthesis of kojic acid derivatives as secondary binding site probes of D-amino acid oxidase.

Johns Hopkins University

Structural, kinetic, and pharmacodynamic mechanisms of D-amino acid oxidase inhibition by small molecules.

Sunovion Pharmaceuticals

Synthesis and SAR study of new thiazole derivatives as vascular adhesion protein-1 (VAP-1) inhibitors for the treatment of diabetic macular edema: part 2.

Astellas Pharma

4-Hydroxypyridazin-3(2H)-one derivatives as novel D-amino acid oxidase inhibitors.

Astellas Pharma

Identification of novel D-amino acid oxidase inhibitors by in silico screening and their functional characterization in vitro.

Kitasato University

Synthesis and SAR study of new thiazole derivatives as vascular adhesion protein-1 (VAP-1) inhibitors for the treatment of diabetic macular edema.

Astellas Pharma

Synthesis and SAR of 1-hydroxy-1H-benzo[d]imidazol-2(3H)-ones as Inhibitors of D-Amino Acid Oxidase.

TBA

The discovery and development of selective 3-fluoro-4-aryloxyallylamine inhibitors of the amine oxidase activity of semicarbazide-sensitive amine oxidase/vascular adhesion protein-1 (SSAO/VAP-1).

Pharmaxis

Biophysical and physicochemical methods differentiate highly ligand-efficient human D-amino acid oxidase inhibitors.

Abbott Healthcare Products

The discovery of fused pyrrole carboxylic acids as novel, potent D-amino acid oxidase (DAO) inhibitors.

Merck Sharp & Dohme

Novel amidino-substituted benzimidazoles: synthesis of compounds and inhibition of dipeptidyl peptidase III.

The Josip Juraj Strossmayer University

3-Amidoquinuclidine derivatives: synthesis of compounds and inhibition of butyrylcholinesterase.

University Of Zagreb