15 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
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Article Title
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Novel bivalent inhibitors with sub-nanomolar affinities towards human glyoxalase I.
Chengdu University
Inhibition by active site directed covalent modification of human glyoxalase I.
University Of Maryland
Synthesis and evaluation of alpha-hydroxythiol esters as antitumor agents and glyoxalase I inhibitors.
TBA
Design and evaluation of azaindole-substituted N-hydroxypyridones as glyoxalase I inhibitors.
Chugai Pharmaceutical
S-(N-aryl-N-hydroxycarbamoyl)glutathione derivatives are tight-binding inhibitors of glyoxalase I and slow substrates for glyoxalase II.
University Of Maryland
Discovery of a new type inhibitor of human glyoxalase I by myricetin-based 4-point pharmacophore.
Tokyo University Of Science
Structural investigation into the inhibitory mechanisms of indomethacin and its analogues towards human glyoxalase I.
Sun Yat-Sen University
Identification of curcumin derivatives as human glyoxalase I inhibitors: A combination of biological evaluation, molecular docking, 3D-QSAR and molecular dynamics simulation studies.
Sun Yat-Sen University
Delphinidin, a dietary anthocyanidin in berry fruits, inhibits human glyoxalase I.
Tokyo University Of Science
Structure-activity relationship of human GLO I inhibitory natural flavonoids and their growth inhibitory effects.
Tokyo University Of Science
Reversal of anticancer drug resistance by COTC based on intracellular glutathione and glyoxalase I.
Keio University
Role of hydrophobic interactions in binding S-(N-aryl/alkyl-N-hydroxycarbamoyl)glutathiones to the active site of the antitumor target enzyme glyoxalase I.
University Of Maryland
Synthesis and activity of gamma-(L-gamma-azaglutamyl)-S-(p-bromobenzyl)-L-cysteinylglycine: a metabolically stable inhibitor of glyoxalase I.
University Of Minnesota