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12 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Novel biguanide-based derivatives scouted as TAAR1 agonists: Synthesis, biological evaluation, ADME prediction and molecular docking studies.EBI
University Of Genoa
Discovery and Characterization of 2-Aminooxazolines as Highly Potent, Selective, and Orally Active TAAR1 Agonists.EBI
Roche Innovation Center Basel
Optimisation of imidazole compounds as selective TAAR1 agonists: discovery of RO5073012.EBI
F. Hoffmann-La Roche
Trace amine-associated receptor 1 is a stereoselective binding site for compounds in the amphetamine class.EBI
Research Triangle Institute
Selective antagonists of mouse trace amine-associated receptor 1 (mTAAR1): discovery of EPPTB (RO5212773).EBI
F. Hoffmann-La Roche
Amiodarone and its putative metabolites fail to activate wild type hTAAR1.EBI
Rti International
Structure-activity correlations for beta-phenethylamines at human trace amine receptor 1.EBI
Rti International
Harnessing Enzymatic Promiscuity in Myxochelin Biosynthesis for the Production of 5-Lipoxygenase Inhibitors.BDB
Hans Knöll Institute