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12 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Selective inhibitors of protein methyltransferases.EBI
Icahn School Of Medicine At Mount Sinai
SAH derived potent and selective EZH2 inhibitors.EBI
Pfizer
Discovery of a selective, substrate-competitive inhibitor of the lysine methyltransferase SETD8.EBI
University Of North Carolina At Chapel Hill
Analogues of the Natural Product Sinefungin as Inhibitors of EHMT1 and EHMT2.EBI
University Of Copenhagen
Selective non-nucleoside inhibitors of human DNA methyltransferases active in cancer including in cancer stem cells.EBI
Sapienza University Of Rome
Discovery and development of potent and selective inhibitors of histone methyltransferase g9a.EBI
Abbvie
Exploiting an allosteric binding site of PRMT3 yields potent and selective inhibitors.EBI
University Of North Carolina At Chapel Hill
Oncoepigenomics: making histone lysine methylation count.EBI
TBA
Optimization of cellular activity of G9a inhibitors 7-aminoalkoxy-quinazolines.EBI
University Of North Carolina At Chapel Hill
Chemical probes for histone-modifying enzymes.EBI
Johns Hopkins University School Of Medicine
Protein lysine methyltransferase G9a inhibitors: design, synthesis, and structure activity relationships of 2,4-diamino-7-aminoalkoxy-quinazolines.EBI
University Of North Carolina At Chapel Hill
Discovery of a 2,4-diamino-7-aminoalkoxyquinazoline as a potent and selective inhibitor of histone lysine methyltransferase G9a.EBI
University Of North Carolina