16 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
PMID
Data
Article Title
Organization
Design and Synthesis of an Investigational Nonapeptide KISS1 Receptor (KISS1R) Agonist, Ac-d-Tyr-Hydroxyproline (Hyp)-Asn-Thr-Phe-azaGly-Leu-Arg(Me)-Trp-NH
Takeda Pharmaceutical
Rational design of triazololipopeptides analogs of kisspeptin inducing a long-lasting increase of gonadotropins.
Umr7247
Physicochemically and pharmacokinetically stable nonapeptide KISS1 receptor agonists with highly potent testosterone-suppressive activity.
Takeda Pharmaceutical
Design, synthesis, and biological evaluation of novel investigational nonapeptide KISS1R agonists with testosterone-suppressive activity.
Takeda Pharmaceutical
Trypsin resistance of a decapeptide KISS1R agonist containing an N¿-methylarginine substitution.
Takeda Pharmaceutical
Serum stability of selected decapeptide agonists of KISS1R using pseudopeptides.
Takeda Pharmaceutical
2-acylamino-4,6-diphenylpyridine derivatives as novel GPR54 antagonists with good brain exposure and in vivo efficacy for plasma LH level in male rats.
Takeda Pharmaceutical
Synthesis and structure-activity relationships of 2-acylamino-4,6-diphenylpyridine derivatives as novel antagonists of GPR54.
Takeda Pharmaceutical
SAR and QSAR studies on the N-terminally acylated pentapeptide agonists for GPR54.
Kyoto University
Metastin (KiSS-1) mimetics identified from peptide structure-activity relationship-derived pharmacophores and directed small molecule database screening.
University Of Minnesota Health Science Center
Neuropeptide FF and Its Receptors: Therapeutic Applications and Ligand Development.
Research Triangle Institute
A new class of pentapeptide KISS1 receptor agonists with hypothalamic-pituitary-gonadal axis activation.
Takeda Pharmaceutical
