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21 articles for AMRI


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDArticle TitlePublishedDeposition
26022843 Discovery of a new chemical series of BRD4(1) inhibitors using protein-ligand docking and structure-guided design. 08-JUN-2015 16-OCT-2016
25050161 Design and synthesis of 4-heteroaryl 1,2,3,4-tetrahydroisoquinolines as triple reuptake inhibitors. 22-JUL-2014 29-MAR-2016
24842618 The design and synthesis of novel SGLT2 inhibitors: C-glycosides with benzyltriazolopyridinone and phenylhydantoin as the aglycone moieties. 02-JUN-2014 11-FEB-2015
24755431 The discovery of diazepinone-based 5-HT3 receptor partial agonists. 09-MAY-2014 09-FEB-2015
23380375 Design, synthesis, and SAR of N-((1-(4-(propylsulfonyl)piperazin-1-yl)cycloalkyl)methyl)benzamide inhibitors of glycine transporter-1. 15-FEB-2013 24-SEP-2013
23084899 4-Phenyl tetrahydroisoquinolines as dual norepinephrine and dopamine reuptake inhibitors. 05-NOV-2012 17-MAY-2013
22503250 Synthesis and SAR studies of imidazo-[1,2-a]-pyrazine Aurora kinase inhibitors with improved off-target kinase selectivity. 07-MAY-2012 07-FEB-2013
20427184 5-Functionalized indazoles as glucocorticoid receptor agonists. 04-MAY-2010 30-DEC-2012
20371178 Synthesis of 7-benzyl-5-(piperidin-1-yl)-6,7,8,9-tetrahydro-3H-pyrazolo[3,4-c][2,7]naphthyridin-1-ylamine and its analogs as bombesin receptor subtype-3 agonists. 20-APR-2010 30-DEC-2012
19846305 Biaryl purine derivatives as potent antiproliferative agents: inhibitors of cyclin dependent kinases. Part I. 05-NOV-2009 26-DEC-2012
19854650 Heterobiaryl purine derivatives as potent antiproliferative agents: inhibitors of cyclin dependent kinases. Part II. 05-NOV-2009 26-DEC-2012
22290076 Epiminocyclohepta[b]indole analogs as 5-HT6 antagonists. 07-FEB-2012 23-JUL-2012
21146988 Novel serotonin type 3 receptor partial agonists for the potential treatment of irritable bowel syndrome. 24-DEC-2010 22-AUG-2011
20951036 Synthesis and SAR of 4-aryl-1-(indazol-5-yl)pyridin-2(1H)ones as MCH-1 antagonists for the treatment of obesity. 08-NOV-2010 14-JUN-2011
20961756 5-(pyridinon-1-yl)indazoles and 5-(furopyridinon-5-yl)indazoles as MCH-1 antagonists. 08-NOV-2010 14-JUN-2011
20952195 Tetrahydrocarboline analogs as MCH-1 antagonists. 08-NOV-2010 14-JUN-2011
20889341 Discovery of 2-substituted benzoxazole carboxamides as 5-HT3 receptor antagonists. 19-OCT-2010 13-JUN-2011
20347296 Synthesis and SAR of heterocyclic carboxylic acid isosteres based on 2-biarylethylimidazole as bombesin receptor subtype-3 (BRS-3) agonists for the treatment of obesity. 20-APR-2010 19-NOV-2010
20022494 2,3-Diaminopyrazines as rho kinase inhibitors. 03-FEB-2010 02-SEP-2010
20079638 Synthesis and structure-activity relationship of substitutions at the C-1 position of Delta9-tetrahydrocannabinol. 15-FEB-2010 01-SEP-2010
19394221 Application of combinatorial biocatalysis for a unique ring expansion of dihydroxymethylzearalenone. 15-MAY-2009 11-JAN-2010