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30 articles for Berlex Biosciences


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDArticle TitlePublishedDeposition
12565961 Structure-activity relationships of substituted benzothiophene-anthranilamide factor Xa inhibitors. 04-FEB-2003 19-MAY-2013
15837303 Solid-phase synthesis of naphthylamidines as factor VIIa/tissue factor inhibitors. 19-APR-2005 02-DEC-2012
12036356 Design, synthesis, and activity of a novel series of factor Xa inhibitors: optimization of arylamidine groups. 30-MAY-2002 26-NOV-2012
10579830 Discovery of novel non-peptide CCR1 receptor antagonists. 17-DEC-1999 13-NOV-2012
19703768 Identification of orally bioavailable, non-amidine inhibitors of Urokinase Plasminogen Activator (uPA). 14-SEP-2009 30-AUG-2010
18590959 Discovery of novel and potent aryl diamines as leukotriene A4 hydrolase inhibitors. 21-JUL-2008 11-JAN-2010
18586492 Synthesis of N-alkyl glycine amides as potent inhibitors of leukotriene A4 hydrolase. 21-JUL-2008 11-JAN-2010
9733479 (Z,Z)-2,7-Bis(4-amidinobenzylidene)cycloheptan-1-one: identification of a highly active inhibitor of blood coagulation factor Xa. 08-OCT-1998 10-NOV-2009
11965377 Design and synthesis of aminophenol-based factor Xa inhibitors. 19-APR-2002 10-NOV-2009
17368901 1-(1,3-Benzodioxol-5-ylmethyl)-3-[4-(1H-imidazol-1-yl)phenoxy]-piperidine analogs as potent and selective inhibitors of nitric oxide formation. 06-APR-2007 10-NOV-2009
17081751 CCR5 receptor antagonists: discovery and SAR study of guanylhydrazone derivatives. 25-DEC-2006 10-NOV-2009
17189688 3-Mercaptopropionic acids as efficacious inhibitors of activated thrombin activatable fibrinolysis inhibitor (TAFIa). 19-FEB-2007 10-NOV-2009
9873451 Solid-phase synthesis of N-substituted amidinophenoxy pyridines as factor XA inhibitors. 04-FEB-1999 10-NOV-2009
12951126 Synthesis and biological evaluation of menthol-based derivatives as inhibitors of plasminogen activator inhibitor-1 (PAI-1). 02-SEP-2003 10-NOV-2009
17336523 The rational design of inhibitors of nitric oxide formation by inducible nitric oxide synthase. 06-APR-2007 10-NOV-2009
14741285 Synthesis and biological evaluation of piperazine-based derivatives as inhibitors of plasminogen activator inhibitor-1 (PAI-1). 26-JAN-2004 10-NOV-2009
17314043 CCR5 receptor antagonists: discovery and SAR of novel 4-hydroxypiperidine derivatives. 13-MAR-2007 10-NOV-2009
17315988 Design, synthesis, and activity of 2-imidazol-1-ylpyrimidine derived inducible nitric oxide synthase dimerization inhibitors. 15-MAR-2007 10-NOV-2009
11965378 Benzimidazole-based fXa inhibitors with improved thrombin and trypsin selectivity. 19-APR-2002 10-NOV-2009
10639283 Synthesis, characterization, and structure-activity relationships of amidine-substituted (bis)benzylidene-cycloketone olefin isomers as potent and selective factor Xa inhibitors. 02-FEB-2000 10-NOV-2009
9733480 Discovery of N-[2-[5-[Amino(imino)methyl]-2-hydroxyphenoxy]-3, 5-difluoro-6-[3-(4, 5-dihydro-1-methyl-1H-imidazol-2-yl)phenoxy]pyridin-4-yl]-N-methylgl y cine (ZK-807834): a potent, selective, and orally active inhibitor of the blood coagulation enzyme factor Xa. 08-OCT-1998 10-NOV-2009
9873520 Design, synthesis, and biological activity of novel purine and bicyclic pyrimidine factor Xa inhibitors. 28-JAN-1999 10-NOV-2009
10346927 Design, synthesis, and activity of 2,6-diphenoxypyridine-derived factor Xa inhibitors. 10-JUN-1999 10-NOV-2009
10853668 Design, synthesis, and in vitro biological activity of indole-based factor Xa inhibitors. 15-NOV-2000 10-NOV-2009
10853669 Design, synthesis, and in vitro biological activity of benzimidazole based factor Xa inhibitors. 15-NOV-2000 10-NOV-2009
18394906 Synthesis of glutamic acid analogs as potent inhibitors of leukotriene A4 hydrolase. 01-MAY-2008 14-SEP-2008
17536795 Thiophene-anthranilamides as highly potent and orally available factor xa inhibitors 28-JUN-2007 08-AUG-2007
17531483 Indolinone based phosphoinositide-dependent kinase-1 (PDK1) inhibitors. Part 1: design, synthesis and biological activity. 15-JUL-2007 02-AUG-2007
15772071 Novel small molecule inhibitors of 3-phosphoinositide-dependent kinase-1. 20-MAY-2005 02-AUG-2007
17544272 Indolinone based phosphoinositide-dependent kinase-1 (PDK1) inhibitors. Part 2: optimization of BX-517. 15-JUL-2007 02-AUG-2007