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261 articles for Burnham Center for Chemical Genomics


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDArticle TitlePublishedDeposition
aid720701 Dose Response confirmation of small molecule inhibitors originally identified via uHTS of Artemis endonuclease activity via a fluorescence intensity assay 29-OCT-2013 08-AUG-2014
aid652002 Dose Response confirmation of uHTS hits for a small molecule Caspase-8 TRAIL sensitizers in a luminescence panel assay 30-JAN-2013 21-JUN-2013
aid652005 Dose response confirmation of small molecule inhibitors of Low Molecular Weight Protein Tyrosine Phosphatase, LMPTP, in an orthogonal absorbance-based assay 01-FEB-2013 21-JUN-2013
aid652006 Dose response confirmation of small molecule inhibitors of Low Molecular Weight Protein Tyrosine Phosphatase, LMPTP, in a fluorescence-based, Lymphoid Phosphatase (PTPN22, LYP-1) selectivity Assay 01-FEB-2013 21-JUN-2013
aid651579 Dose Response Confirmation of SKN-1 Inhibitor hits via a heat-shock counterscreen assay 12-SEP-2012 20-JUN-2013
aid651565 Dose-response confirmation of uHTS inhibitor hits of Sentrin-Specific Protease 8 in a Caspase-3 Fluorescence assay 05-SEP-2012 20-JUN-2013
aid651570 Dose response validation of uHTS Gli-SUFU antagonist hits in a Wnt3a luminescent reporter assay 07-SEP-2012 20-JUN-2013
aid651563 Dose ResponseConfirmation of SKN-1 Inhibitor hits in a fluorescence ratio assay - Set 2 05-SEP-2012 20-JUN-2013
aid651709 Dose response confirmation of uHTS inhibitor hits from NadD in a Colorimetric assay - Set 2 26-OCT-2012 20-JUN-2013
aid651684 Dose response confirmation of small molecule activators of alpha dystroglycan glycosylation 23-OCT-2012 20-JUN-2013
aid651639 Dose Response confirmation of uHTS hits for small molecule antagonists of the CRF-binding protein and CRF-R2 receptor complex in 384 well format 12-OCT-2012 20-JUN-2013
aid651650 Dose Response confirmation of small molecule modulators of the interaction between CendR and NRP-1 in a panel assay 18-OCT-2012 20-JUN-2013
aid651581 Dose response confirmation of uHTS identification of HIF-2a Inhibitors in a luminesence assay 12-SEP-2012 20-JUN-2013
aid651559 Dose-response confirmation of uHTS inhibitor hits of Sentrin-Specific Protease 8 using a kinetic assay with Nedd8 Protein Substrate 04-SEP-2012 20-JUN-2013
aid651559 Dose-response confirmation of uHTS inhibitor hits of Sentrin-Specific Protease 8 using a kinetic assay with Nedd8 Protein Substrate 04-SEP-2012 20-JUN-2013
aid651675 SAR analysis of small molecule activators of alpha dystroglycan glycosylation 22-OCT-2012 20-JUN-2013
aid651594 Dose Response counterscreen of small molecule antagonists of the CXCR6 receptor using a CXCR5 receptor luminescent beta-arrestin assay 21-SEP-2012 20-JUN-2013
aid651693 Dose response confirmation of small molecule inhibitors of the catalytic domain of the SUMO protease, SENP1 in a FRET assay 23-OCT-2012 20-JUN-2013
aid651697 Dose response confirmation of small molecule inhibitors of the catalytic domain of the SUMO protease, SENP1 in a kinetic FRET assay 24-OCT-2012 20-JUN-2013
aid651700 Dose response confirmation of small molecule inhibitors of Low Molecular Weight Protein Tyrosine Phosphatase, LMPTP, via a fluorescence intensity assay 25-OCT-2012 20-JUN-2013
aid624241 Dose Response selectivity of inhibitors of STriatal-Enriched Phosphatase (STEP) in the Lymphoid Phosphatase (PTPN22) Inhibition Assay 30-MAY-2012 25-JUN-2012
aid624207 Dose response orthogonal assay of uHTS small molecule inhibitors of Striatal-Enriched Phosphatase via a colorimetric intensity assay. 29-MAY-2012 25-JUN-2012
aid602374 Dose Response selectivity of inhibitors of STriatal-Enriched Phosphatase (STEP) in the dual-specificity protein-tyrosine phosphatase VHR Inhibition Assay 13-MAR-2012 19-JUN-2012
aid602369 Dose Response validation of uHTS RPN11 inhibitor hits using a Thrombin Fluorescence Polarization assay 12-MAR-2012 19-JUN-2012
aid602378 SAR analysis of small molecule inhibitors of tim23-1: a luminescent tim10-1 yeast counterscreen. 13-MAR-2012 19-JUN-2012
aid602380 SAR analysis of small molecule inhibitors of tim23-1: a luminescent TIM10 yeast counterscreen. 13-MAR-2012 19-JUN-2012
aid602386 Dose response confirmation of DNMT1 inhibitors in a Fluorescent Molecular Beacon assay 13-MAR-2012 19-JUN-2012
aid602461 SAR analysis of small molecule inhibitors of Apaf-1 using a LZ-Caspase-9/Caspase-3 Fluorescent Selectivity assay - Set 2 22-MAR-2012 19-JUN-2012
aid602464 Dose response confirmation of uHTS antagonist hits from Gli-SUFU in a luminescent reporter assay 22-MAR-2012 19-JUN-2012
aid602469 SAR analysis of small molecule Activators of Apaf-1 in a Fluorescent assay - set 2 22-MAR-2012 19-JUN-2012
aid602460 SAR analysis of small molecule Inhibitors of Apaf-1 in a Fluorescent assay - set 2 22-MAR-2012 19-JUN-2012
aid602372 Dose response confirmation of uHTS small molecule inhibitors of Striatal-Enriched Phosphatase via a fluorescence intensity assay 12-MAR-2012 19-JUN-2012
aid602367 Dose Response selectivity of inhibitors of Striatal-Enriched Phosphatase (STEP) in a SHP2 (PTPN11) Inhibition Assay 12-MAR-2012 19-JUN-2012
aid624089 SAR analysis of small molecule inhibitors of APOBEC3A DNA Deaminase via a fluorescence-based single-stranded DNA deaminase assay - Set 2 12-APR-2012 19-JUN-2012
aid624087 SAR analysis of small molecule inhibitors of APOBEC3G DNA Deaminase via a fluorescence-based single-stranded DNA deaminase assay - Set 2 12-APR-2012 19-JUN-2012
aid602471 SAR analysis of small molecule activators of Apaf-1 using a LZ-Caspase-9/Caspase-3 Fluorescent Selectivity assay - Set 2 22-MAR-2012 19-JUN-2012
aid602375 SAR analysis of small molecule inhibitors of tim23-1 yeast via a luminescent assay 13-MAR-2012 19-JUN-2012
aid602473 Dose Response confirmation of uHTS hits for small molecule agonists of the CRF-binding protein and CRF-R2 receptor complex 22-MAR-2012 19-JUN-2012
aid602260 Dose-response secondary confirmation of microRNA-mediated mRNA deadenylation inhibitors by fluoresence polarization assay using Cy5 labeled peptide 14-FEB-2012 19-JUN-2012
aid602259 Dose-response confirmation of microRNA-mediated mRNA deadenylation inhibitors by fluoresence polarization assay 14-FEB-2012 19-JUN-2012
aid602368 Dose response confirmation of uHTS RPN11 inhibitor hits in a Fluorescence Polarization assay 12-MAR-2012 19-JUN-2012
aid602136 SAR analysis of small molecule inhibitors of APOBEC3G DNA Deaminase via a fluorescence-based single-stranded DNA deaminase assay 16-DEC-2011 18-JUN-2012
aid588574 Dose response confirmation of uHTS hits for Apaf-1 using a LZ-Caspase-9/Caspase-3 Fluorescent Selectivity assay 25-OCT-2011 06-JAN-2012
aid588586 Dose response counterscreen of uHTS hits for ATG4B inhibitors in a Phospholipase A2 assay Set 2 20-OCT-2011 06-JAN-2012
aid588554 Dose Response confirmation of uHTS Activators of the Apaf-1 Pathway in Fluorescent format 18-OCT-2011 06-JAN-2012
aid588603 SAR analysis of small molecule activators of the MazEF TA System via a fluorescence-based single-stranded RNase assay 21-OCT-2011 06-JAN-2012
aid588601 SAR Analysis of small molecule inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay - Set 2 21-OCT-2011 06-JAN-2012
aid588592 Dose Response validation of Activators of Apaf-1 using a Fluorescent Interference Counterscreen assay 20-OCT-2011 06-JAN-2012
aid588584 Dose response confirmation of the uHTS fluorescent assay for identification of inhibitors of ATG4B Set 2 20-OCT-2011 06-JAN-2012
aid588400 Dose response counterscreen of uHTS hits for ATG4B inhibitors in a Phospholipase A2 assay 22-SEP-2011 05-JAN-2012
aid588502 Dose response confirmation uHTS hits for MazEF TA System activators via a fluorescence-based single-stranded RNase assay counterscreen 12-OCT-2011 05-JAN-2012
aid588538 Dose Response validation of Inhibitors of Apaf-1 using a Fluorescent Interference Counterscreen assay 17-OCT-2011 05-JAN-2012
aid588359 SAR analysis counterscreen of small molecule antagonists of the CCR6 receptor using an APJ receptor luminescent beta-arrestin assay 14-SEP-2011 05-JAN-2012
aid588481 Dose response confirmation uHTS hits for MazEF TA System activators via a fluorescence-based single-stranded RNase assay 11-OCT-2011 05-JAN-2012
aid588524 Dose response confirmation of uHTS hits for Apaf-1 in a Fluorescent assay 25-OCT-2011 05-JAN-2012
aid540269 Dose Response orthogonal kinetic assay utilizing the direct detection of NADPH for uHTS small molecule inhibitors of Plasmodium falciparum Glucose-6-phosphate dehydrogenase 18-JUL-2011 04-JAN-2012
aid540334 SAR analysis of small molecule antagonists of the CCR6 receptor: a luminescent beta-arrestin assay 08-AUG-2011 04-JAN-2012
aid540252 Dose Response orthogonal assay utilizing the direct end-point detection of NADPH for uHTS small molecule inhibitors of Plasmodium falciparum Glucose-6-phosphate dehydrogenase 14-JUL-2011 04-JAN-2012
aid540288 SAR VHR1 Fluorescent Assay for In Vitro dose response studies Set 3 23-JUL-2011 04-JAN-2012
aid540297 Dose Response confirmation of uHTS hits for Scp-1 phosphatase using a colorimetric assay 23-JUL-2011 04-JAN-2012
aid504763 Dose Response confirmation of inhibitors of hexokinase domain containing I (HKDC1) in the hexokinase 1 selectivity assay 13-MAY-2011 04-AUG-2011
aid504792 Human Glucose-6-Phosphate Dehydrogenase Dose Response Selectivity Assay for Inhibitors of Plasmodium falciparum Glucose-6-Phosphate Dehydrogenase 03-JUN-2011 04-AUG-2011
aid504765 Dose Response confirmation of uHTS small molecule inhibitors of Plasmodium falciparum Glucose-6-phosphate dehydrogenase via a fluorescence intensity assay 18-MAY-2011 04-AUG-2011
aid504762 Dose Response confirmation of activators of hexokinase domain containing I (HKDC1) in the hexokinase 1 selectivity assay 13-MAY-2011 04-AUG-2011
aid504544 Dose Response confirmation of uHTS small molecule inhibitors of tim10-1: a luminescent tim23-1 yeast counterscreen. 23-MAR-2011 03-AUG-2011
aid504549 Dose Response confirmation of Image-Based HTS for Selective Agonists for NTR1 23-MAR-2011 03-AUG-2011
aid504593 Dose Response confirmation of Inhibitors of Mdm2/MdmX interaction in luminescent format 28-MAR-2011 03-AUG-2011
aid504712 HTS Dose response counterscreen for assays utilizing the enzyme, beta-galactosidase - Set 3 29-APR-2011 03-AUG-2011
aid504723 Dose Response confirmation of APOBEC3A DNA Deaminase Inhibitors via a A3G counterscreen 05-MAY-2011 03-AUG-2011
aid504728 Dose Response confirmation of small molecule antagonists of the CCR6 receptor: a luminescent beta-arrestin assay 05-MAY-2011 03-AUG-2011
aid504729 Dose Response confirmation of inhibitors of hexokinase domain containing I (HKDC1) 06-MAY-2011 03-AUG-2011
aid504730 Dose Response confirmation of activators of hexokinase domain containing I (HKDC1) 06-MAY-2011 03-AUG-2011
aid504756 Dose response confirmation of the uHTS fluorescent assay for identification of inhibitors of ATG4B. 13-MAY-2011 03-AUG-2011
aid504657 Dose Response confirmation of uHTS small molecule inhibitors of tim23-1: a luminescent tim10-1 yeast counterscreen. 13-APR-2011 03-AUG-2011
aid504669 Dose Response confirmation of Inhibitors of Mdm2/MdmX interaction using a Brca1/Bard1 BiLC Counterscreen assay 14-APR-2011 03-AUG-2011
aid504672 Dose Response confirmation of uHTS small molecule inhibitors of tim23-1: a luminescent TIM10 yeast counterscreen. 14-APR-2011 03-AUG-2011
aid504719 Dose Response confirmation of small molecule APOBEC3G DNA Deaminase Inhibitors via a fluorescence-based single-stranded DNA deaminase assay 04-MAY-2011 03-AUG-2011
aid504722 Dose Response confirmation of APOBEC3G DNA Deaminase Inhibitors via a A3A counterscreen 05-MAY-2011 03-AUG-2011
aid504724 Dose Response confirmation of small molecule APOBEC3A DNA Deaminase Inhibitors via a fluorescence-based single-stranded DNA deaminase assay 05-MAY-2011 03-AUG-2011
aid504689 Dose Response confirmation of UBC13 Polyubiquitin Inhibitors using a Bfl-1 counterscreen 20-APR-2011 03-AUG-2011
aid493155 Dose Response confirmation of uHTS for the identification of UBC13 Polyubiquitin Inhibitors via a TR-FRET Assay 03-FEB-2011 02-AUG-2011
aid493003 Dose Response confirmation of uHTS small molecule inhibitors of tim10-1 yeast via a luminescent assay 21-DEC-2010 02-AUG-2011
aid493182 Dose Response confirmation of uHTS for the identification of UBC13 Polyubiquitin Inhibitors via a TR-FRET Assay reconfirm 10-FEB-2011 02-AUG-2011
aid488879 Dose Response confirmation of uHTS inhibitors of Mouse Intestinal Alkaline Phosphatase using Placental Alkaline Phosphatase 25-OCT-2010 01-AUG-2011
aid488880 Dose Response confirmation of uHTS activators of Mouse Intestinal Alkaline Phosphatase using Tissue Nonspecific Alkaline Phosphatase. 25-OCT-2010 01-AUG-2011
aid488882 Dose Response confirmation of uHTS inhibitors of Human Intestinal Alkaline Phosphatase using Tissue Nonspecific Alkaline Phosphatase. 25-OCT-2010 01-AUG-2011
aid488884 SAR Selectivity Analysis of small molecule inhibitors of PEST using pCAP in a fluorescence assay 25-OCT-2010 01-AUG-2011
aid488886 Dose Response confirmation of uHTS activators of Human Intestinal Alkaline Phosphatase using Tissue Nonspecific Alkaline Phosphatase. 25-OCT-2010 01-AUG-2011
aid488888 Dose Response confirmation of uHTS activators of Human Intestinal Alkaline Phosphatase using Placental Alkaline Phosphatase 25-OCT-2010 01-AUG-2011
aid488892 Dose Response confirmation of uHTS inhibitors of Human Intestinal Alkaline Phosphatase using Placental Alkaline Phosphatase 25-OCT-2010 01-AUG-2011
aid488901 Dose Response confirmation of inhibitors of Sentrin-specific proteases (SENPs) using a Caspase-3 Selectivity assay 26-OCT-2010 01-AUG-2011
aid488923 Dose Response confirmation of compounds that inhibit HePTP 26-OCT-2010 01-AUG-2011
aid488925 SAR analysis of Antagonists of the Kappa Opioid Receptor (KOR) using an Image-Based Assay - Set 4 26-OCT-2010 01-AUG-2011
aid488935 SAR analysis of small molecule antagonists of the kappa opioid receptor via a luminescent beta-arrestin assay - Set 6 26-OCT-2010 01-AUG-2011
aid488957 SAR analysis of Antagonists of IAP-family anti-apoptotic proteins - Set 2 27-OCT-2010 01-AUG-2011
aid485278 SAR analysis of antagonists of the Cannabinoid Receptor 2 using an Image-Based Assay - Set 3 27-SEP-2010 01-AUG-2011
aid485282 SAR analysis of agonists of the Cannabinoid Receptor 1 using an Image-Based Assay - Set 4 27-SEP-2010 01-AUG-2011
aid488783 Dose Response concentration confirmation of uHTS hits from a small molecule activators of mouse intestinal alkaline phosphatase via a luminescent assay 14-OCT-2010 01-AUG-2011
aid488793 Dose Response confirmation of uHTS hits from a small molecule inhibitors of human intestinal alkaline phosphatase via a luminescent assay - Set 2 14-OCT-2010 01-AUG-2011
aid488799 Dose Response confirmation of uHTS for the identification of inhibitors of NALP3 in yeast using a luminescent assay 15-OCT-2010 01-AUG-2011
aid488863 Dose Response confirmation of inhibitors of NALP1 in yeast using a Caspase-1-ASC counter screen. 21-OCT-2010 01-AUG-2011
aid488865 Dose Response screen for agonists of Angiotensin II Receptor Type 1 to assess selectivity of uHTS small molecule agonists hits of the APJ receptor 22-OCT-2010 01-AUG-2011
aid488873 Dose Response confirmation of uHTS activators of Mouse Intestinal Alkaline Phosphatase using Human Intestinal Alkaline Phosphatase 25-OCT-2010 01-AUG-2011
aid488874 Dose Response confirmation of uHTS inhibitors of Human Intestinal Alkaline Phosphatase using Mouse Intestinal Alkaline Phosphatase 25-OCT-2010 01-AUG-2011
aid488903 Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay 26-OCT-2010 01-AUG-2011
aid488906 Dose Response confirmation of uHTS inhibitors of Mouse Intestinal Alkaline Phosphatase using Tissue Nonspecific Alkaline Phosphatase. 26-OCT-2010 01-AUG-2011
aid488920 Dose Response confirmation of inhibitors of Sentrin-specific proteases (SENPs) using a Luminescent Interference Counterscreen assay 26-OCT-2010 01-AUG-2011
aid488921 Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 6 (SENP6) using a Luminescent assay 26-OCT-2010 01-AUG-2011
aid488963 SAR analysis of Antagonists of XIAP-Bir3 domain of IAP-family anti-apoptotic proteins - Set 2 28-OCT-2010 01-AUG-2011
aid488987 SAR Analysis for the identification of Selective Antagonists of ERK1/2 Activity in GPR35-Overexpressing U2OS Cells - Set 2 03-NOV-2010 01-AUG-2011
aid463217 SAR Analysis for the identification of Selective Antagonists of ERK1/2 Activity in GPR35-Overexpressing U2OS Cells 10-SEP-2010 01-AUG-2011
aid463227 SAR analysis of Antagonists of the GPR35 Receptor using an Image-Based Assay - Set 5 12-NOV-2010 01-AUG-2011
aid463228 SAR Analysis of Selective Antagonists of GPR55 using an Image-Based Assay - Set 3 16-SEP-2010 01-AUG-2011
aid485277 SAR analysis of agonists of the Cannabinoid Receptor 2 using an Image-Based Assay - Set 3 27-SEP-2010 01-AUG-2011
aid485283 SAR analysis of Antagonists of the GPR35 Receptor using an Image-Based Assay - Set 6 27-SEP-2010 01-AUG-2011
aid485285 SAR analysis of antagonists of the Cannabinoid Receptor 1 using an Image-Based Assay - Set 4 27-SEP-2010 01-AUG-2011
aid485286 SAR analysis of Agonists of the GPR35 Receptor using an Image-Based Assay - Set 4 27-SEP-2010 01-AUG-2011
aid485287 SAR Analysis of Selective Antagonists of GPR55 using an Image-Based Assay - Set 4 27-SEP-2010 01-AUG-2011
aid485352 HTS Dose response counterscreen for assays utilizing the enzyme, beta-galactosidase - Set 2 05-OCT-2010 01-AUG-2011
aid488748 Dose Response confirmation of uHTS hits from a small molecule agonists of the APJ receptor via a luminescent beta-arrestin assay 08-OCT-2010 01-AUG-2011
aid488785 Dose Response confirmation of uHTS hits from a small molecule inhibitors of mouse intestinal alkaline phosphatase via a luminescent assay 14-OCT-2010 01-AUG-2011
aid488800 Dose Response confirmation of inhibitors of NALP3 in yeast using a Caspase-1-ASC counter screen 15-OCT-2010 01-AUG-2011
aid488817 Dose Response concentration confirmation of uHTS hits from a small molecule activators of human intestinal alkaline phosphatase via a luminescent assay - Set 2 18-OCT-2010 01-AUG-2011
aid488819 SAR analysis of Antagonists of the Kappa Opioid Receptor (KOR) using an Image-Based Assay - Set 3 18-OCT-2010 01-AUG-2011
aid488822 SAR Analysis of Agonists of the MOR Receptor using an Image-Based Assay - Set 3 19-OCT-2010 01-AUG-2011
aid488824 SAR Analysis of Agonists of the DOR Receptor using an Image-Based Assay - Set 3 19-OCT-2010 01-AUG-2011
aid488826 SAR analysis of small molecule antagonists of the kappa opioid receptor via a luminescent beta-arrestin assay - Set 5 19-OCT-2010 01-AUG-2011
aid488831 SAR Analysis of Antagonists of the DOR Receptor using an Image-Based Assay - Set 3 19-OCT-2010 01-AUG-2011
aid488833 SAR analysis of Agonists of the Kappa Opioid Receptor (KOR) using an Image-Based Assay-Set 3 19-OCT-2010 01-AUG-2011
aid488842 SAR Analysis of Antagonists of the MOR Receptor using an Image-Based Assay - Set 3 20-OCT-2010 01-AUG-2011
aid488860 Dose Response confirmation of uHTS for the identification of inhibitors of NALP1 in yeast using a luminescent assay 21-OCT-2010 01-AUG-2011
aid488861 Dose Response Confirmation of compounds that inhibit VHR1 in Fluorescent Assay 21-OCT-2010 01-AUG-2011
aid488869 SAR LYP1 Fluorescent Assay using OMFP substrate for In Vitro dose response studies - Set 4 22-OCT-2010 01-AUG-2011
aid488876 Dose Response confirmation of uHTS inhibitors of Mouse Intestinal Alkaline Phosphatase using Human Intestinal Alkaline Phosphatase 25-OCT-2010 01-AUG-2011
aid488871 SAR LYP1 Fluorescent Assay using pCAP substrate for In Vitro dose response studies - Set 4 25-OCT-2010 01-AUG-2011
aid488878 Dose Response confirmation of uHTS activators of Mouse Intestinal Alkaline Phosphatase using Placental Alkaline Phosphatase 25-OCT-2010 01-AUG-2011
aid488875 Dose Response confirmation of uHTS activators of Human Intestinal Alkaline Phosphatase using Mouse Intestinal Alkaline Phosphatase 25-OCT-2010 01-AUG-2011
aid449727 SAR LYP1 Fluorescent Assay using pCAP substrate for In Vitro dose response studies - Set 3 07-JUL-2010 31-JUL-2011
aid435027 Dose Response confirmation of uHTS hits from a small molecule inhibitors of LYP via a fluorescence intensity assay using pCAP substrate 30-JUN-2010 31-JUL-2011
aid435024 Dose Response confirmation of uHTS hits from a small molecule inhibitors of LYP via a fluorescence intensity assay - Set 2 29-JUN-2010 31-JUL-2011
aid463135 Dose Response confirmation of uHTS hits from a small molecule inhibitors of human intestinal alkaline phosphatase via a luminescent assay 25-AUG-2010 31-JUL-2011
aid449737 SAR analysis of small molecule agonists of the kappa opioid receptor via a luminescent beta-arrestin assay - Set 3 08-JUL-2010 31-JUL-2011
aid463214 Dose Response screen for antagonists of Angiotensin II Receptor Type 1 to assess selectivity of uHTS small molecule antagonists hits of the APJ receptor 08-SEP-2010 31-JUL-2011
aid463120 Dose Response concentration confirmation of uHTS hits from a small molecule activators of human intestinal alkaline phosphatase via a luminescent assay 24-AUG-2010 31-JUL-2011
aid463105 SAR analysis of small molecule antagonists of the kappa opioid receptor via a luminescent beta-arrestin assay - Set 4 18-AUG-2010 31-JUL-2011
aid449733 SAR analysis of compounds that inhibit VHR1, Fluorescent Assay - Set 2 07-JUL-2010 31-JUL-2011
aid449736 SAR analysis of compounds that inhibit HePTP - Set 2 08-JUL-2010 31-JUL-2011
aid449726 SAR LYP1 Fluorescent Assay using OMFP substrate for In Vitro dose response studies - Set 3 06-JUL-2010 31-JUL-2011
aid435032 Dose Response confirmation of HTS hits from an HePTP Fluorescent Assay using OMFP substrate - Set 2 01-JUL-2010 31-JUL-2011
aid435029 SAR analysis of compounds that inhibit Human Immunodeficiency Virus Fusion, cell-cell fusion assay 01-JUL-2010 31-JUL-2011
aid435018 SAR analysis for the identification of translation initiation inhibitors (PABP) 25-JUN-2010 31-JUL-2011
aid435011 SAR analysis for the identification of translation initiation inhibitors (eIF4H) 22-JUN-2010 31-JUL-2011
aid434980 SAR analysis of small molecule inhibitors of Mint-PDZ and N-type Ca2+ channel carboxyl-terminal peptide association using HTRF - Set 2 07-JUN-2010 30-JUL-2011
aid434967 SAR analysis of compounds that inhibit Human Immunodeficiency Virus Fusion. 03-JUN-2010 30-JUL-2011
aid434981 SAR analysis of small molecule antagonists of the kappa opioid receptor via a luminescent beta-arrestin assay - Set 3 07-JUN-2010 30-JUL-2011
aid434924 SAR analysis of Agonists of the GPR35 Receptor using an Image-Based Assay - Set 3 20-MAY-2010 29-JUL-2011
aid434929 SAR analysis of antagonists of the Cannabinoid Receptor 1 using an Image-Based Assay - Set 3 20-MAY-2010 29-JUL-2011
aid434925 SAR analysis of Antagonists of the GPR35 Receptor using an Image-Based Assay - Set 4 20-MAY-2010 29-JUL-2011
aid434922 SAR analysis of antagonists of the Cannabinoid Receptor 2 using an Image-Based Assay - Set 2 20-MAY-2010 29-JUL-2011
aid434928 SAR analysis of agonists of the Cannabinoid Receptor 2 using an Image-Based Assay - Set 2 20-MAY-2010 29-JUL-2011
aid2798 SAR analysis of compounds that inhibit NOD1 - Set 3 04-MAY-2010 12-JUL-2011
aid2793 SAR analysis of NF-kappaB dependent luciferase using DAP as an inducer - Set 2 28-APR-2010 12-JUL-2011
aid2792 SAR analysis of NF-kappaB dependent luciferase using PMA/Ionomycin as an inducer - 2 28-APR-2010 12-JUL-2011
aid2789 SAR analysis of NF-kappaB dependent luciferase using Doxorucibin as an inducer - Set 2 28-APR-2010 12-JUL-2011
aid2801 SAR analysis of inhibitors of TNFa specific NF-kB induction - Set 3 04-MAY-2010 12-JUL-2011
aid2799 SAR analysis of compounds that inhibit NOD2 - Set 3 04-MAY-2010 12-JUL-2011
aid2505 SAR analysis of GM-Tri-DAP induced IL-8 secretion in MCF-7/NOD1 cells - Set 2 10-MAR-2010 11-JUL-2011
aid2504 SAR analysis of Tumor necrosis factor alpha (TNF-alpha) induced IL-8 secretion in MCF-7/NOD1 cells - Set 2 10-MAR-2010 11-JUL-2011
aid2500 SAR analysis of small molecule agonists of the kappa opioid receptor via a luminescent beta-arrestin assay - Set 2 12-NOV-2010 11-JUL-2011
aid2492 SAR Analysis of Agonists of the MOR Receptor using an Image-Based Assay - Set 2 06-MAR-2010 11-JUL-2011
aid2497 SAR analysis of Agonists of the Kappa Opioid Receptor (KOR) using an Image-Based Assay - Set 2 08-MAR-2010 11-JUL-2011
aid2493 SAR Analysis of Agonists of the DOR Receptor using an Image-Based Assay - Set 2 06-MAR-2010 11-JUL-2011
aid2491 SAR analysis of Antagonists of the Kappa Opioid Receptor (KOR) using an Image-Based Assay - Set 2 06-MAR-2010 11-JUL-2011
aid2489 SAR analysis of small molecule inhibitors of Mint-PDZ and N-type Ca2+ channel carboxyl-terminal peptide association using HTRF 05-MAR-2010 11-JUL-2011
aid2682 SAR LYP1 Fluorescent Assay using pCAP substrate for In Vitro dose response studies - Set 2 25-MAR-2010 11-JUL-2011
aid2503 SAR analysis of Muramyl dipeptide (MDP) induced IL-8 secretion in MCF-7/NOD2 cells - Set 2 09-MAR-2010 11-JUL-2011
aid2485 HTS dose response assay for identification of inhibitors of TNFa-specific NF-kB induction 05-MAR-2010 11-JUL-2011
aid2483 SAR analysis of inhibitors of TNFa specific NF-kB induction - Set 2 05-MAR-2010 11-JUL-2011
aid2480 SAR analysis of Antagonists of the GPR35 Receptor using an Image-Based Assay - Set 2 05-MAR-2010 11-JUL-2011
aid2686 SAR LYP1 Fluorescent Assay using OMFP substrate for In Vitro dose response studies - Set 2 25-MAR-2010 11-JUL-2011
aid2466 SAR analysis of compounds that inhibit NOD1 - Set 2 06-MAY-2010 11-JUL-2011
aid2475 SAR analysis of compounds that inhibit NOD2 - Set 2 05-APR-2010 11-JUL-2011
aid2348 SAR analysis of Antagonists of the Kappa Opioid Receptor (KOR) using an Image-Based Assay 11-FEB-2010 10-JUL-2011
aid2356 HTS Image-Based Screen for Antagonists of the DOR Receptor 18-MAR-2010 10-JUL-2011
aid2359 SAR analysis of Agonists of the Kappa Opioid Receptor (KOR) using an Image-Based Assay 12-FEB-2010 10-JUL-2011
aid2370 SAR Analysis of Agonists of the DOR Receptor using an Image-Based Assay 16-FEB-2010 10-JUL-2011
aid2420 SAR Analysis of Antagonists of the MOR Receptor using an Image-Based Assay 24-FEB-2010 10-JUL-2011
aid2397 SAR Analysis of Selective Antagonists of GPR55 using an Image-Based Assay 16-SEP-2010 10-JUL-2011
aid2338 SAR analysis of Antagonists of the GPR35 Receptor using an Image-Based Assay 05-FEB-2010 10-JUL-2011
aid2343 HTS Image-Based Screen for Agonists of the DOR Receptor 09-FEB-2010 10-JUL-2011
aid2352 SAR Analysis of Agonists of the MOR Receptor using an Image-Based Assay 12-FEB-2010 10-JUL-2011
aid2357 SAR Analysis of Antagonists of the DOR Receptor using an Image-Based Assay 12-FEB-2010 10-JUL-2011
aid1961 Image-based HTS for Selective Agonists of GPR55 17-JUN-2010 09-JUL-2011
aid2012 uHTS fluorescence polarization assay for the identification of translation initiation inhibitors (eIF4H) 11-DEC-2009 09-JUL-2011
aid2058 Image-Based HTS for Selective Antagonists of GPR35 15-JUN-2010 09-JUL-2011
aid2006 uHTS HTRF assay for identification of inhibitors of SUMOylation 22-JAN-2010 09-JUL-2011
aid2013 Image-Based HTS for Selective Antagonists for GPR55 15-JUN-2010 09-JUL-2011
aid2014 uHTS fluorescence polarization assay for the identification of translation initiation inhibitors (PABP) 11-DEC-2009 09-JUL-2011
aid1817 uHTS identification of small molecule antagonists of the binding of Siah-1 and a peptide ligand via a fluorescence polarization assay. 12-NOV-2009 09-JUL-2011
aid1778 uHTS identification of small molecule antagonists of the kappa opioid receptor via a luminescent beta-arrestin assay 14-SEP-2009 09-JUL-2011
aid1654 uHTS absorbance assay for the identification of compounds that inhibit VHR1. 09-JUL-2009 09-JUL-2011
aid1779 uHTS identification of small molecule inhibitors of LYP via a fluorescence intensity assay 12-NOV-2009 09-JUL-2011
aid2264 SAR analysis of NF-kB dependent luciferase using DAP as an inducer 15-JAN-2010 09-JUL-2011
aid2337 SAR analysis of inhibitors of TNFa specific NF-kB induction revised 04-FEB-2010 09-JUL-2011
aid2334 SAR analysis of compounds that inhibit NOD2 revised 13-APR-2010 09-JUL-2011
aid2333 SAR analysis of compounds that inhibit NOD1 revised 03-FEB-2010 09-JUL-2011
aid2285 SAR analysis of small molecule antagonists of the kappa opioid receptor via a luminescent beta-arrestin assay 22-JAN-2010 09-JUL-2011
aid2284 SAR analysis of small molecule agonists of the kappa opioid receptor via a luminescent beta-arrestin assay 22-JAN-2010 09-JUL-2011
aid2073 Homogeneous Time-Resolved Fluorescence Resonance Energy Transfer (HTRF) Assay 09-NOV-2009 09-JUL-2011
aid1578 uHTS luminescence assay for the identification of compounds that inhibit NOD1 17-FEB-2010 08-JUL-2011
aid696 Luminescent assay for HTS discovery of chemical activators of placental alkaline phosphatase 24-APR-2007 08-JUL-2011
aid2141 HTS TR-FRET-based dose response confirmatory assay for Siah-1 15-NOV-2009 05-JUN-2011
aid2140 SAR LYP1 Fluorescent Assay using OMFP substrate for In Vitro dose response studies 15-NOV-2009 05-JUN-2011
aid2136 HTS Image-Based Screen for Selective Antagonists of the KOR Receptor 12-NOV-2009 05-JUN-2011
aid2135 SAR LYP1 Fluorescent Assay using pCAP substrate for In Vitro dose response studies 12-NOV-2009 05-JUN-2011
aid2134 HTS HePTP Fluorescent Assay using OMFP substrate for In Vitro dose response studies 12-NOV-2009 05-JUN-2011
aid2133 HTS Image-Based Screen for Selective Agonists of the KOR Receptor 12-NOV-2009 05-JUN-2011
aid2127 HTS fluorescence polarization-based dose response confirmatory screen for the Siah-1 primary assay utilizing an alternative fluorophore, fluorescein-labeled plectin 12-NOV-2009 05-JUN-2011
aid2126 LYP1 Fluorescent Assay using OMFP substrate for In Vitro dose response studies. 12-NOV-2009 05-JUN-2011
aid2070 MOA VHR1 Fluorescent secondary assay for identification of redox-state modulating compounds 28-OCT-2009 05-JUN-2011
aid2091 uHTS Homogeneous Terbium Time-Resolved Fluorescence Resonance Energy Transfer (HTRF) Assay 30-OCT-2009 05-JUN-2011
aid2068 MOA HePTP Fluorescent secondary assay for identification of redox-state modulating compounds 28-OCT-2009 05-JUN-2011
aid2018 AlphaScreen confirmatory assay for validation of inhibitors of SUMOylation 21-JAN-2010 05-JUN-2011
aid2001 uHTS luminescence assay for the identification of compounds that inhibit NOD2 in MDP treated cells 19-JAN-2010 05-JUN-2011
aid568 High Throughput Screening Assay for Hsc70 Inhibitors 16-APR-2007 04-JUN-2011
aid521 HTS Discovery of Chemical Inhibitors of HePTP, a Leukemia Target 11-FEB-2008 04-JUN-2011
aid1659 SAR assay for compounds activating TNAP in the presence of 100 mM DEA performed in a luminescence assay 20-AUG-2009 31-MAY-2011
aid1878 Fluorescent assay for identification of compounds that inhibit VHR1 18-JUL-2009 31-MAY-2011
aid1957 SAR VHR1 Fluorescent Assay for In Vitro dose response studies 02-NOV-2009 29-MAY-2011
aid1941 SAR assay for compounds inhibiting TNAP in the absence of phosphate acceptor performed in a luminescent assay 12-NOV-2010 29-MAY-2011
aid1966 HTS Dose response counterscreen for assays utilizing the enzyme, b-galactosidase 05-OCT-2009 29-MAY-2011
aid1958 SAR VHR1 absorbance Assay for In Vitro dose response studies. 29-SEP-2009 29-MAY-2011
aid1536 Confirmation of compounds inhibiting phosphomannose isomerase (PMI) via a fluorescence intensity assay using a high concentration of mannose 6-phosphate. 05-MAR-2009 28-MAY-2011
aid1535 Confirmation of compounds inhibiting phosphomannose isomerase (PMI) via a fluorescence intensity assay. 12-NOV-2010 28-MAY-2011
aid1514 Counter Screen using XIAP-Bir3 of the Chemical Antagonists of IAP-family anti-apoptotic proteins confirmation assay 29-JAN-2009 28-MAY-2011
aid1512 Luminescent assay for HTS discovery of chemical inhibitors of placental alkaline phosphatase confirmation 11-JUN-2009 28-MAY-2011
aid1655 Counter screen SAR assay for PMM2 inhibitors via a fluorescence intensity assay 12-NOV-2010 28-MAY-2011
aid1056 SAR analysis of an In Vitro TNAP Dose Response Luminescent Assay 12-NOV-2010 28-MAY-2011
aid1077 Fluorescent secondary assay for dose-response confirmation of chemical inhibitors of HePTP 31-OCT-2009 28-MAY-2011
aid1666 SAR assay for compounds that inhibit PHOSPHO1 12-NOV-2010 28-MAY-2011
aid518 TNAP luminescent HTS assay 05-FEB-2008 27-MAY-2011
aid779 Counter Screen for Placental Alkaline Phosphatase-based Assays Positives 11-FEB-2008 27-MAY-2011
aid1755 SAR analysis of compounds that potentiate TRAIL-induced apoptosis in MDA-MB-435 cells. 13-MAY-2009 25-MAY-2011
aid1752 SAR analysis of compounds that potentiate TRAIL-induced apoptosis in PPC-1 cells. 13-MAY-2009 25-MAY-2011
aid1750 SAR analysis of Antagonists of XIAP-Bir3 domain of IAP-family anti-apoptotic proteins 05-NOV-2009 25-MAY-2011
aid1749 SAR analysis of Antagonists of IAP-family anti-apoptotic proteins 04-NOV-2009 25-MAY-2011
aid1450 SAR assay for compounds activating TNAP in the absence of phosphate acceptor performed in a luminescent assay 12-NOV-2010 21-MAY-2011
aid1449 Chemical Antagonists of IAP-family anti-apoptotic proteins confirmation 27-JAN-2009 21-MAY-2011
aid1052 MKP-3 in vitro secondary assay for identification of irreversible and slow-binding inhibitors 28-FEB-2008 17-MAY-2011
aid1072 In Vitro Hsp70 Dose Response Fluorescence Polarization Assay for SAR Study 03-MAR-2008 17-MAY-2011
aid786 TR-FRET secondary assay for HTS discovery of chemical inhibitors of Hsp70 11-FEB-2008 11-MAY-2011
aid748 High Throughput Fluorescence Polarization Screen for Bcl-B Phenotype Converters 21-NOV-2008 06-MAY-2011
aid690 Luminescent assay for HTS discovery of chemical inhibitors of placental alkaline phosphatase 23-APR-2007 30-APR-2011
aid1220 HTS identification of compounds inhibiting phosphomannose isomerase (PMI) via a fluorescence intensity assay using a high concentration of mannose 6-phosphate 03-MAR-2009 24-NOV-2009
aid432 HTS discovery of chemical inhibitors of anti-apoptotic protein Bfl-1 09-FEB-2008 24-NOV-2009
aid583 High Throughput Screening Assay for Hsp70 Inhibitors 11-FEB-2008 25-SEP-2009
aid1055 In Vitro MKP-3 Dose Response Assay for SAR Study 28-FEB-2008 25-SEP-2009
aid1560 Confirmation of compounds inhibiting the binding between the RUNX1 Runt domain and CBFb-SMMHC via a fluorescence resonance energy transfer (FRET) assay 18-MAR-2009 24-JUL-2009
aid1550 Confirmation of compounds inhibiting the binding between the RUNX1 Runt domain and CBFbeta-SMMHC via a time resolved fluorescence resonance energy transfer (TR-FRET) assay. 13-MAR-2009 24-JUL-2009
aid1434 uHTS identification of compounds inhibiting the binding between the RUNX1 Runt domain and CBFbeta-SMMHC via a fluorescence resonance energy transfer (FRET) assay. 23-JAN-2009 24-JUL-2009
aid1438 Identification of compounds inhibiting the binding between the RUNX1 Runt domain and CBFb-SMMHC via a time resolved fluorescence resonance energy transfer (TR-FRET) assay. 23-JAN-2009 18-JUN-2009