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28 articles for CNRS


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDArticle TitlePublishedDeposition
27676471 Further investigation of Paprotrain: Towards the conception of selective and multi-targeted CNS kinase inhibitors. 29-NOV-2016 02-SEP-2018
27214508 Straightforward synthesis of 2,4,6-trisubstituted 1,3,5-triazine compounds targeting cysteine cathepsins K and S. 04-OCT-2016 17-JUL-2018
26778612 New MKLP-2 inhibitors in the paprotrain series: Design, synthesis and biological evaluations. 02-FEB-2016 05-JUN-2017
26752095 Design and synthesis of calindol derivatives as potent and selective calcium sensing receptor agonists. 02-FEB-2016 04-JUN-2017
22998443 Selectivity, cocrystal structures, and neuroprotective properties of leucettines, a family of protein kinase inhibitors derived from the marine sponge alkaloid leucettamine B. 08-NOV-2012 17-MAY-2013
22483635 Chemical synthesis and biological evaluation of triazole derivatives as inhibitors of InhA and antituberculosis agents. 30-APR-2012 07-FEB-2013
18993066 Beta-C-glycosiduronic acids and beta-C-glycosyl compounds: new PTP1B inhibitors. 25-NOV-2008 18-DEC-2012
16913701 N1-Benzoyl-N2-[1-(1-naphthyl)ethyl]-trans-1,2-diaminocyclohexanes: Development of 4-chlorophenylcarboxamide (calhex 231) as a new calcium sensing receptor ligand demonstrating potent calcilytic activity. 17-AUG-2006 08-DEC-2012
10673095 First enantiospecific synthesis of a 3,4-dihydroxy-L-glutamic acid [(3S,4S)-DHGA], a new mGluR1 agonist. 07-MAR-2000 01-OCT-2012
8450829 Mouse 5-hydroxytryptamine5A and 5-hydroxytryptamine5B receptors define a new family of serotonin receptors: cloning, functional expression, and chromosomal localization. XX-XXX-1993 10-FEB-2012
8394987 Molecular cloning of a mammalian serotonin receptor that activates adenylate cyclase. XX-XXX-1993 09-FEB-2012
21435752 New potent human acetylcholinesterase inhibitors in the tetracyclic triterpene series with inhibitory potency on amyloid β aggregation. 02-MAY-2011 06-DEC-2011
1464308 The mouse 5HT5 receptor reveals a remarkable heterogeneity within the 5HT1D receptor family. XX-XXX-1992 10-NOV-2011
19161318 A Dimeric sesquiterpenoid from a Malaysian Meiogyne as a new inhibitor of Bcl-xL/BakBH3 domain peptide interaction. 11-MAR-2010 26-AUG-2010
19572612 Cytotoxic pentacyclic triterpenoids from Combretum sundaicum and Lantana camara as inhibitors of Bcl-xL/BakBH3 domain peptide interaction. 01-SEP-2009 26-AUG-2010
18922697 Synthesis of triazole-linked beta-C-glycosyl dimers as inhibitors of PTP1B. 05-NOV-2008 11-JAN-2010
18467107 Substituted benzyl-pyrimidines targeting thymidine monophosphate kinase of Mycobacterium tuberculosis: synthesis and in vitro anti-mycobacterial activity. 05-JUN-2008 11-JAN-2010
7932576 Structure-activity study of neuropeptide FF: contribution of N-terminal regions to affinity and activity. 23-NOV-1994 10-NOV-2009
10964567 Structural basis for isotype selectivity of the human retinoic acid nuclear receptor. 08-SEP-2000 28-SEP-2009
19334715 Design, synthesis, and biological evaluation of new 5-HT4 receptor agonists: application as amyloid cascade modulators and potential therapeutic utility in Alzheimer's disease. 23-APR-2009 07-JUN-2009
19237285 Benzimidazolone-based serotonin 5-HT1A or 5-HT7R ligands: synthesis and biological evaluation. 15-MAR-2009 07-JUN-2009
11906289 Toward an optimal joint recognition of the S1' subsites of endothelin converting enzyme-1 (ECE-1), angiotensin converting enzyme (ACE), and neutral endopeptidase (NEP). 28-MAR-2002 19-APR-2008
17927165 Toward Potent Ghrelin Receptor Ligands Based on Trisubstituted 1,2,4-Triazole Structure. 2. Synthesis and Pharmacological in Vitro and in Vivo Evaluations. 15-NOV-2007 10-DEC-2007
17902635 New potent acetylcholinesterase inhibitors in the tetracyclic triterpene series. 01-NOV-2007 15-NOV-2007
15026054 Meridianins, a new family of protein kinase inhibitors isolated from the ascidian Aplidium meridianum. 05-APR-2004 26-AUG-2006
9839013 Potent acetylcholinesterase inhibitors: design, synthesis, and structure-activity relationships of bis-interacting ligands in the galanthamine series. 00-OCT-1998 31-JUL-2006
15830466 Synthesis and anticancer activity of new pyrrolocarbazoles and pyrrolo-beta-carbolines. 15-MAR-2005 21-JAN-2006
10998059 Paullones are potent inhibitors of glycogen synthase kinase-3beta and cyclin-dependent kinase 5/p25. 00-OCT-2000 12-JAN-2006