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17 articles for Clinical Research Institute of Montreal

The following articles (labelled with PubMed ID or TBD) are for your review
PMIDArticle TitlePublishedDeposition
27676089 A Cyclic Tetrapeptide ("Cyclodal") and Its Mirror-Image Isomer Are Both High-Affinityµ Opioid Receptor Antagonists. 13-OCT-2016 20-JUL-2018
25129170 'Carba'-carfentanil (trans isomer): aµ opioid receptor (MOR) partial agonist with a distinct binding mode. 29-8 -2014 29-OCT-2016
22325949 Novel TIPP (H-Tyr-Tic-Phe-Phe-OH) analogues displaying a wide range of efficacies at thed opioid receptor. Discovery of two highly potent and selectived opioid agonists. 21-FEB-2012 17-MAY-2013
20218625 "Carba"-analogues of fentanyl are opioid receptor agonists. 01-APR-2010 30-DEC-2012
11543672 [2',6'-Dimethyltyrosine]dynorphin A(1-11)-NH2 analogues lacking an N-terminal amino group: potent and selective kappa opioid antagonists. 06-SEP-2001 25-NOV-2012
8164255 Cyclic beta-casomorphin analogues with mixed mu agonist/delta antagonist properties: synthesis, pharmacological characterization, and conformational aspects. 24-MAY-1994 29-OCT-2012
8230106 TIPP[psi]: a highly potent and stable pseudopeptide delta opioid receptor antagonist with extraordinary delta selectivity. 26-NOV-1993 25-OCT-2012
11121615 Synthesis and in vitro opioid activity profiles of DALDA analogues. XX-XXX-2000 25-APR-2012
19827750 Agonist vs antagonist behavior of delta opioid peptides containing novel phenylalanine analogues in place of Tyr(1). 05-NOV-2009 29-AUG-2010
2822930 Structure-activity relationships of cyclic opioid peptide analogues containing a phenylalanine residue in the 3-position. 09-DEC-1987 10-NOV-2009
10479285 The opioid mu agonist/delta antagonist DIPP-NH(2)[Psi] produces a potent analgesic effect, no physical dependence, and less tolerance than morphine in rats. 14-OCT-1999 10-NOV-2009
1656045 Conformational restriction of the phenylalanine residue in a cyclic opioid peptide analogue: effects on receptor selectivity and stereospecificity. 18-NOV-1991 10-NOV-2009
2537427 Dermorphin analogues carrying an increased positive net charge in their"message" domain display extremely high mu opioid receptor selectivity. 06-APR-1989 10-NOV-2009
11212101 Stereospecific synthesis of (2S)-2-methyl-3-(2',6'-dimethyl-4'-hydroxyphenyl)-propionic acid (Mdp) and its incorporation into an opioid peptide. 09-FEB-2001 10-NOV-2009
1331451 Conformationally restricted deltorphin analogues. 27-NOV-1992 10-NOV-2009
15324897 A novel cyclic enkephalin analogue with potent opioid antagonist activity. 24-AUG-2004 10-NOV-2009
17315860 Dicarba analogues of the cyclic enkephalin peptides H-Tyr-c[D-Cys-Gly-Phe-D(or L)-Cys]NH(2) retain high opioid activity. 15-MAR-2007 10-NOV-2009