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45 articles for Emory University

The following articles (labelled with PubMed ID or TBD) are for your review
PMIDArticle TitlePublishedDeposition
US9428478 Piperazine derivatives, compositions, and uses related thereto 30-AUG-2016 21-AUG-2017
26525866 A novel class of negative allosteric modulators of NMDA receptor function. 06-NOV-2015 24-MAY-2017
26456805 Synthesis, binding affinity, radiolabeling, and microPET evaluation of 4-(2-substituted-4-substituted)-8-(dialkylamino)-6-methyl-1-substituted-3,4-dihydropyrido[2,3-b]pyrazin-2(1H)-ones as ligands for brain corticotropin-releasing factor type-1 (CRF1) receptors. 31-OCT-2015 15-DEC-2016
26191361 Pyrazolo-Piperidines Exhibit Dual Inhibition of CCR5/CXCR4 HIV Entry and Reverse Transcriptase. 20-7 -2015 19-NOV-2016
26005525 Design and Validation of FRESH, a Drug Discovery Paradigm Resting on Robust Chemical Synthesis. 25-MAY-2015 11-OCT-2016
US9205085 Tricyclic amino containing compounds for treatment or prevention of symptoms associated with endocrine dysfunction 08-DEC-2015 03-OCT-2016
27427228 Structural Basis for KDM5A Histone Lysine Demethylase Inhibition by Diverse Compounds. 21-JUL-2016 01-SEP-2016
24937185 Development of second generation EP2 antagonists with high selectivity. 28-JUN-2014 12-FEB-2015
24512267 Design, synthesis, and structure-activity relationship of a novel series of GluN2C-selective potentiators. 27-MAR-2014 07-FEB-2015
23978650 Investigation of an F-18 oxytocin receptor selective ligand via PET imaging. 06-SEP-2013 13-APR-2014
23909910 Structure-activity relationships and pharmacophore model of a noncompetitive pyrazoline containing class of GluN2C/GluN2D selective antagonists. 22-AUG-2013 13-APR-2014
23550937 Monocarbonyl curcumin analogues: heterocyclic pleiotropic kinase inhibitors that mediate anticancer properties. 09-MAY-2013 24-SEP-2013
18092818 Comparison of the structural properties of the active site cavities of human and rat monoamine oxidase A and B in their soluble and membrane-bound forms. 15-JAN-2008 18-MAR-2013
22425346 Synthesis and evaluation of C-11, F-18 and I-125 small molecule radioligands for detecting oxytocin receptors. 06-APR-2012 07-FEB-2013
20597489 Synthesis, fluorine-18 radiolabeling, and biological evaluation of N-((E)-4-fluorobut-2-en-1-yl)-2beta-carbomethoxy-3beta-(4'-halophenyl)nortropanes: candidate radioligands for in vivo imaging of the brain dopamine transporter with positron emission tomography. 05-AUG-2010 01-JAN-2013
18800760 Enantiomeric propanolamines as selective N-methyl-D-aspartate 2B receptor antagonists. 19-SEP-2008 19-DEC-2012
19067522 Synthesis, radiosynthesis, and biological evaluation of carbon-11 and fluorine-18 labeled reboxetine analogues: potential positron emission tomography radioligands for in vivo imaging of the norepinephrine transporter. 02-JAN-2009 18-DEC-2012
18472268 Synthesis, fluorine-18 radiolabeling, and in vitro characterization of 1-iodophenyl-N-methyl-N-fluoroalkyl-3-isoquinoline carboxamide derivatives as potential PET radioligands for imaging peripheral benzodiazepine receptor. 05-JUN-2008 16-DEC-2012
17983754 Synthesis, in vitro characterization, and radiolabeling of reboxetine analogs as potential PET radioligands for imaging the norepinephrine transporter. 01-FEB-2008 15-DEC-2012
10072683 Synthesis and biological evaluation of 2',3'-didehydro-2',3'- dideoxy-5-fluorocytidine (D4FC) analogues: discovery of carbocyclic nucleoside triphosphates with potent inhibitory activity against HIV-1 reverse transcriptase. 11-MAR-1999 13-NOV-2012
14744476 Milnacipran: a comparative analysis of human monoamine uptake and transporter binding affinity. 01-XXX-2004 29-MAY-2012
12065700 Biochemistry and pharmacology of epitope-tagged alpha(1)-adrenergic receptor subtypes. XX-XXX-2002 09-MAY-2012
12232544 [Second generation SSRIS: human monoamine transporter binding profile of escitalopram and R-fluoxetine]. XX-XXX-0 09-MAY-2012
10755640 18F-labeled FECNT: a selective radioligand for PET imaging of brain dopamine transporters. XX-XXX-2000 17-APR-2012
21105715 Dipyrimidine amines: a novel class of chemokine receptor type 4 antagonists with high specificity. 17-DEC-2010 23-MAR-2012
9400006 Neurotransmitter receptor and transporter binding profile of antidepressants and their metabolites. XX-XXX-1997 01-MAR-2012
9131252 Pharmacology and functions of metabotropic glutamate receptors. XX-XXX-1997 25-FEB-2012
20684595 Quinazolin-4-one derivatives: A novel class of noncompetitive NR2C/D subunit-selective N-methyl-D-aspartate receptor antagonists. 05-AUG-2010 20-MAR-2011
19648014 Synthesis, structural activity-relationships, and biological evaluation of novel amide-based allosteric binding site antagonists in NR1A/NR2B N-methyl-D-aspartate receptors. 21-AUG-2009 31-AUG-2010
19053782 Synthesis, radiosynthesis, and biological evaluation of fluorine-18-labeled 2beta-carbo(fluoroalkoxy)-3beta-(3'-((Z)-2-haloethenyl)phenyl)nortropanes: candidate radioligands for in vivo imaging of the serotonin transporter with positron emission tomography. 18-DEC-2008 11-JAN-2010
19053775 Structural and mechanistic studies of mofegiline inhibition of recombinant human monoamine oxidase B. 18-DEC-2008 11-JAN-2010
17958344 Discovery of small molecule CXCR4 antagonists. 08-NOV-2007 11-NOV-2009
18085744 Synthesis and in vivo evaluation of halogenated N,N-dimethyl-2-(2'-amino-4'-hydroxymethylphenylthio)benzylamine derivatives as PET serotonin transporter ligands. 17-JAN-2008 11-NOV-2009
16574411 Synthesis and evaluation of two 18F-labeled imidazo[1,2-a]pyridine analogues as potential agents for imaging beta-amyloid in Alzheimer's disease. 24-APR-2006 10-NOV-2009
10691690 Synthesis, biodistribution, and primate imaging of fluorine-18 labeled 2beta-carbo-1'-fluoro-2-propoxy-3beta-(4-chlorophenyl)tr opanes. Ligands for the imaging of dopamine transporters by positron emission tomography. 16-MAR-2000 10-NOV-2009
12620070 Synthesis and characterization of iodine-123 labeled 2beta-carbomethoxy-3beta-(4'-((Z)-2-iodoethenyl)phenyl)nortropane. A ligand for in vivo imaging of serotonin transporters by single-photon-emission tomography. 06-MAR-2003 10-NOV-2009
14971892 Synthesis, radiosynthesis, and biological evaluation of carbon-11 and iodine-123 labeled 2beta-carbomethoxy-3beta-[4'-((Z)-2-haloethenyl)phenyl]tropanes: candidate radioligands for in vivo imaging of the serotonin transporter. 19-FEB-2004 10-NOV-2009
15974579 Synthesis, in vitro characterization, and radiolabeling of N,N-dimethyl-2-(2'-amino-4'-substituted-phenylthio)benzylamines: potential candidates as selective serotonin transporter radioligands. 24-JUN-2005 10-NOV-2009
16451060 Evaluation of carbon-11-labeled 2beta-carbomethoxy-3beta-[4'-((Z)-2-iodoethenyl)phenyl]nortropane as a potential radioligand for imaging the serotonin transporter by PET. 02-FEB-2006 10-NOV-2009
16784855 Synthesis and monoamine transporter affinity of front bridged tricyclic 3beta-(4'-halo or 4'-methyl)phenyltropanes bearing methylene or carbomethoxymethylene on the bridge to the 2beta-position. 31-JUL-2006 10-NOV-2009
17154506 Synthesis, radiosynthesis, and biological evaluation of carbon-11 labeled 2beta-carbomethoxy-3beta-(3'-((Z)-2-haloethenyl)phenyl)nortropanes: candidate radioligands for in vivo imaging of the serotonin transporter with positron emission tomography. 12-DEC-2006 10-NOV-2009
17446069 Synthesis and biological evaluation of 2beta,3alpha-(substituted phenyl)nortropanes as potential norepinephrine transporter imaging agents. 14-MAY-2007 10-NOV-2009
17705359 Synthesis and in vivo evaluation of fluorine-18 and iodine-123 labeled 2beta-carbo(2-fluoroethoxy)-3beta-(4'-((Z)-2-iodoethenyl)phenyl)nortropane as a candidate serotonin transporter imaging agent. 13-SEP-2007 10-NOV-2009
15027867 Inactivation of purified human recombinant monoamine oxidases A and B by rasagiline and its analogues. 25-MAR-2004 12-SEP-2006
15710600 Demonstration of isoleucine 199 as a structural determinant for the selective inhibition of human monoamine oxidase B by specific reversible inhibitors. 22-APR-2005 12-SEP-2006