BindingDB logo
myBDB logout

45 articles for Emory University


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDArticle TitlePublishedDeposition
US9428478 Piperazine derivatives, compositions, and uses related thereto 30-AUG-2016 21-AUG-2017
26525866 A novel class of negative allosteric modulators of NMDA receptor function. 06-NOV-2015 24-MAY-2017
26456805 Synthesis, binding affinity, radiolabeling, and microPET evaluation of 4-(2-substituted-4-substituted)-8-(dialkylamino)-6-methyl-1-substituted-3,4-dihydropyrido[2,3-b]pyrazin-2(1H)-ones as ligands for brain corticotropin-releasing factor type-1 (CRF1) receptors. 31-OCT-2015 15-DEC-2016
26191361 Pyrazolo-Piperidines Exhibit Dual Inhibition of CCR5/CXCR4 HIV Entry and Reverse Transcriptase. 20-7 -2015 19-NOV-2016
26005525 Design and Validation of FRESH, a Drug Discovery Paradigm Resting on Robust Chemical Synthesis. 25-MAY-2015 11-OCT-2016
US9205085 Tricyclic amino containing compounds for treatment or prevention of symptoms associated with endocrine dysfunction 08-DEC-2015 03-OCT-2016
27427228 Structural Basis for KDM5A Histone Lysine Demethylase Inhibition by Diverse Compounds. 21-JUL-2016 01-SEP-2016
24937185 Development of second generation EP2 antagonists with high selectivity. 28-JUN-2014 12-FEB-2015
24512267 Design, synthesis, and structure-activity relationship of a novel series of GluN2C-selective potentiators. 27-MAR-2014 07-FEB-2015
23978650 Investigation of an F-18 oxytocin receptor selective ligand via PET imaging. 06-SEP-2013 13-APR-2014
23909910 Structure-activity relationships and pharmacophore model of a noncompetitive pyrazoline containing class of GluN2C/GluN2D selective antagonists. 22-AUG-2013 13-APR-2014
23550937 Monocarbonyl curcumin analogues: heterocyclic pleiotropic kinase inhibitors that mediate anticancer properties. 09-MAY-2013 24-SEP-2013
18092818 Comparison of the structural properties of the active site cavities of human and rat monoamine oxidase A and B in their soluble and membrane-bound forms. 15-JAN-2008 18-MAR-2013
22425346 Synthesis and evaluation of C-11, F-18 and I-125 small molecule radioligands for detecting oxytocin receptors. 06-APR-2012 07-FEB-2013
20597489 Synthesis, fluorine-18 radiolabeling, and biological evaluation of N-((E)-4-fluorobut-2-en-1-yl)-2beta-carbomethoxy-3beta-(4'-halophenyl)nortropanes: candidate radioligands for in vivo imaging of the brain dopamine transporter with positron emission tomography. 05-AUG-2010 01-JAN-2013
18800760 Enantiomeric propanolamines as selective N-methyl-D-aspartate 2B receptor antagonists. 19-SEP-2008 19-DEC-2012
19067522 Synthesis, radiosynthesis, and biological evaluation of carbon-11 and fluorine-18 labeled reboxetine analogues: potential positron emission tomography radioligands for in vivo imaging of the norepinephrine transporter. 02-JAN-2009 18-DEC-2012
18472268 Synthesis, fluorine-18 radiolabeling, and in vitro characterization of 1-iodophenyl-N-methyl-N-fluoroalkyl-3-isoquinoline carboxamide derivatives as potential PET radioligands for imaging peripheral benzodiazepine receptor. 05-JUN-2008 16-DEC-2012
17983754 Synthesis, in vitro characterization, and radiolabeling of reboxetine analogs as potential PET radioligands for imaging the norepinephrine transporter. 01-FEB-2008 15-DEC-2012
10072683 Synthesis and biological evaluation of 2',3'-didehydro-2',3'- dideoxy-5-fluorocytidine (D4FC) analogues: discovery of carbocyclic nucleoside triphosphates with potent inhibitory activity against HIV-1 reverse transcriptase. 11-MAR-1999 13-NOV-2012
14744476 Milnacipran: a comparative analysis of human monoamine uptake and transporter binding affinity. 01-XXX-2004 29-MAY-2012
12065700 Biochemistry and pharmacology of epitope-tagged alpha(1)-adrenergic receptor subtypes. XX-XXX-2002 09-MAY-2012
12232544 [Second generation SSRIS: human monoamine transporter binding profile of escitalopram and R-fluoxetine]. XX-XXX-0 09-MAY-2012
10755640 18F-labeled FECNT: a selective radioligand for PET imaging of brain dopamine transporters. XX-XXX-2000 17-APR-2012
21105715 Dipyrimidine amines: a novel class of chemokine receptor type 4 antagonists with high specificity. 17-DEC-2010 23-MAR-2012
9400006 Neurotransmitter receptor and transporter binding profile of antidepressants and their metabolites. XX-XXX-1997 01-MAR-2012
9131252 Pharmacology and functions of metabotropic glutamate receptors. XX-XXX-1997 25-FEB-2012
20684595 Quinazolin-4-one derivatives: A novel class of noncompetitive NR2C/D subunit-selective N-methyl-D-aspartate receptor antagonists. 05-AUG-2010 20-MAR-2011
19648014 Synthesis, structural activity-relationships, and biological evaluation of novel amide-based allosteric binding site antagonists in NR1A/NR2B N-methyl-D-aspartate receptors. 21-AUG-2009 31-AUG-2010
19053782 Synthesis, radiosynthesis, and biological evaluation of fluorine-18-labeled 2beta-carbo(fluoroalkoxy)-3beta-(3'-((Z)-2-haloethenyl)phenyl)nortropanes: candidate radioligands for in vivo imaging of the serotonin transporter with positron emission tomography. 18-DEC-2008 11-JAN-2010
19053775 Structural and mechanistic studies of mofegiline inhibition of recombinant human monoamine oxidase B. 18-DEC-2008 11-JAN-2010
17958344 Discovery of small molecule CXCR4 antagonists. 08-NOV-2007 11-NOV-2009
18085744 Synthesis and in vivo evaluation of halogenated N,N-dimethyl-2-(2'-amino-4'-hydroxymethylphenylthio)benzylamine derivatives as PET serotonin transporter ligands. 17-JAN-2008 11-NOV-2009
16574411 Synthesis and evaluation of two 18F-labeled imidazo[1,2-a]pyridine analogues as potential agents for imaging beta-amyloid in Alzheimer's disease. 24-APR-2006 10-NOV-2009
10691690 Synthesis, biodistribution, and primate imaging of fluorine-18 labeled 2beta-carbo-1'-fluoro-2-propoxy-3beta-(4-chlorophenyl)tr opanes. Ligands for the imaging of dopamine transporters by positron emission tomography. 16-MAR-2000 10-NOV-2009
12620070 Synthesis and characterization of iodine-123 labeled 2beta-carbomethoxy-3beta-(4'-((Z)-2-iodoethenyl)phenyl)nortropane. A ligand for in vivo imaging of serotonin transporters by single-photon-emission tomography. 06-MAR-2003 10-NOV-2009
14971892 Synthesis, radiosynthesis, and biological evaluation of carbon-11 and iodine-123 labeled 2beta-carbomethoxy-3beta-[4'-((Z)-2-haloethenyl)phenyl]tropanes: candidate radioligands for in vivo imaging of the serotonin transporter. 19-FEB-2004 10-NOV-2009
15974579 Synthesis, in vitro characterization, and radiolabeling of N,N-dimethyl-2-(2'-amino-4'-substituted-phenylthio)benzylamines: potential candidates as selective serotonin transporter radioligands. 24-JUN-2005 10-NOV-2009
16451060 Evaluation of carbon-11-labeled 2beta-carbomethoxy-3beta-[4'-((Z)-2-iodoethenyl)phenyl]nortropane as a potential radioligand for imaging the serotonin transporter by PET. 02-FEB-2006 10-NOV-2009
16784855 Synthesis and monoamine transporter affinity of front bridged tricyclic 3beta-(4'-halo or 4'-methyl)phenyltropanes bearing methylene or carbomethoxymethylene on the bridge to the 2beta-position. 31-JUL-2006 10-NOV-2009
17154506 Synthesis, radiosynthesis, and biological evaluation of carbon-11 labeled 2beta-carbomethoxy-3beta-(3'-((Z)-2-haloethenyl)phenyl)nortropanes: candidate radioligands for in vivo imaging of the serotonin transporter with positron emission tomography. 12-DEC-2006 10-NOV-2009
17446069 Synthesis and biological evaluation of 2beta,3alpha-(substituted phenyl)nortropanes as potential norepinephrine transporter imaging agents. 14-MAY-2007 10-NOV-2009
17705359 Synthesis and in vivo evaluation of fluorine-18 and iodine-123 labeled 2beta-carbo(2-fluoroethoxy)-3beta-(4'-((Z)-2-iodoethenyl)phenyl)nortropane as a candidate serotonin transporter imaging agent. 13-SEP-2007 10-NOV-2009
15027867 Inactivation of purified human recombinant monoamine oxidases A and B by rasagiline and its analogues. 25-MAR-2004 12-SEP-2006
15710600 Demonstration of isoleucine 199 as a structural determinant for the selective inhibition of human monoamine oxidase B by specific reversible inhibitors. 22-APR-2005 12-SEP-2006