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32 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
26947959 35 Synthesis, structural characterization, docking, lipophilicity and cytotoxicity of 1-[(1R)-1-(6-fluoro-1,3-benzothiazol-2-yl)ethyl]-3-alkyl carbamates, novel acetylcholinesterase and butyrylcholinesterase pseudo-irreversible inhibitors.EBI University of Pardubice
26632651 70 Novel Tacrine-Benzofuran Hybrids as Potent Multitarget-Directed Ligands for the Treatment of Alzheimer's Disease: Design, Synthesis, Biological Evaluation, and X-ray Crystallography.EBI China Pharmaceutical University
26363872 19 Synthesis and structure-activity relationship study of benzofuran-based chalconoids bearing benzylpyridinium moiety as potent acetylcholinesterase inhibitors.EBI Alzahra University
26260334 28 Galantamine derivatives with indole moiety: Docking, design, synthesis and acetylcholinesterase inhibitory activity.EBI Medical University of Sofia
25017625 45 Synthesis and cholinesterase inhibition of cativic acid derivatives.EBI Universidad Nacional del Sur
24835788 28 Preparation, anticholinesterase activity and molecular docking of new lupane derivatives.EBI Universidad Nacional del Sur
18538575 3 Petrosamine, a potent anticholinesterase pyridoacridine alkaloid from a Thai marine sponge Petrosia n. sp.EBI Mahidol University
18479118 113 Exploiting protein fluctuations at the active-site gorge of human cholinesterases: further optimization of the design strategy to develop extremely potent inhibitors.EBI Universit£ di Siena
17944454 34 First gallamine-tacrine hybrid: design and characterization at cholinesterases and the M2 muscarinic receptor.EBI University of Bonn
15139762 133 Interaction of cycloSal-pronucleotides with cholinesterases from different origins. A structure-activity relationship.EBI University of Hamburg
10052979 45 Aminopyridazines as acetylcholinesterase inhibitors.EBI Universit£ Louis Pasteur
8978837 60 Structure-based alignment and comparative molecular field analysis of acetylcholinesterase inhibitors.EBI University of North Carolina
8893840 12 The simulated binding of (+/-)-2,3-dihydro-5,6-dimethoxy-2-[[1-(phenylmethyl)-4-piperidinyl]meth yl] -1H-inden-1-one hydrochloride (E2020) and related inhibitors to free and acylated acetylcholinesterases and corresponding structure-activity analyses.EBI Eisai Co., Ltd.
19726199 30 Rational design and synthesis of highly potent anti-acetylcholinesterase activity huperzine A derivatives.EBI The Chinese Academy of Sciences
 5 m-Alkyl, α,α,α-trifluoroacetophenones: A new class of potent transition state analog inhibitors of acetylcholinesteraseEBI TBA
17317172 9 Methyl 2-(2-(4-formylphenoxy)acetamido)-2-substituted acetate derivatives: a new class of acetylcholinesterase inhibitors.EBI Sun Yat-sen University
14584959 55 Molecular docking studies of natural cholinesterase-inhibiting steroidal alkaloids from Sarcococca saligna.EBI University of Innsbruck
12729674 6 Synthesis, anticholinesterase activity and structure-activity relationships of m-Aminobenzoic acid derivatives.EBI Instituto Politécnico Nacional
9871563 31 Synthesis and activity studies of N-[omega-N'-(adamant-1'-yl)aminoalkyl]- 2-(4'-dimethylaminophenyl)acetamides: in the search of selective inhibitors for the different molecular forms of acetylcholinesterase.EBI Istituto di Strutturistica Chimica G. Giacomello
26322521 6 Inhibition and Allosteric Regulation of Monomeric Phosphoenolpyruvate Carboxykinase by 3-Mercaptopicolinic Acid.BDB The University of Kansas Medical Center
18849971 56 Targeted polypharmacology: discovery of dual inhibitors of tyrosine and phosphoinositide kinases.BDB University of California, San Francisco
18942826 19 Inhibitor Scaffolds for 2-Oxoglutarate-Dependent Histone Lysine Demethylases.BDB University of Oxford
18227510 8 The T790M mutation in EGFR kinase causes drug resistance by increasing the affinity for ATP.BDB Harvard Medical School
17846131 15 Small-molecule scaffolds for CYP51 inhibitors identified by high-throughput screening and defined by X-ray crystallography.BDB University of California at San Francisco
18473434 57 Novel inhibitors of the v-raf murine sarcoma viral oncogene homologue B1 (BRAF) based on a 2,6-disubstituted pyrazine scaffold.BDB Cancer Research UK Centre for Cancer Therapeutics
18925736 19 Structure-activity relationship studies of phenanthridine-based Bcl-XL inhibitors.BDB A*STAR
18793847 33 Design and synthesis of 2-amino-pyrazolopyridines as Polo-like kinase 1 inhibitors.BDB Sunesis Pharmaceuticals