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24 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
28609101 49 Design, Synthesis, and Evaluation of Thiazolidine-2,4-dione Derivatives as a Novel Class of Glutaminase Inhibitors.EBI National Health Research Institutes
28174105 9 Physapubescin, a natural withanolide as a kidney-type glutaminase (KGA) inhibitor.EBI Huazhong University of Science and Technology
27200176 22 Allosteric Glutaminase Inhibitors Based on a 1,4-Di(5-amino-1,3,4-thiadiazol-2-yl)butane Scaffold.EBI Johns Hopkins University
26985303 12 Glutaminase GLS1 Inhibitors as Potential Cancer Treatment.EBI Therachem Research Medilab (India) Pvt. Ltd.
26988803 32 Design and evaluation of novel glutaminase inhibitors.EBI University of Pittsburgh
23151085 29 Design, synthesis, and pharmacological evaluation of bis-2-(5-phenylacetamido-1,2,4-thiadiazol-2-yl)ethyl sulfide 3 (BPTES) analogs as glutaminase inhibitors.EBI Johns Hopkins University
30148361 7 Overview of the Development of Glutaminase Inhibitors: Achievements and Future Directions.EBI China Pharmaceutical University
31474484 20 GAC inhibitors with a 4-hydroxypiperidine spacer: Requirements for potency.EBI University of Pittsburgh
30543285 27 Novel 1,3,4-Selenadiazole-Containing Kidney-Type Glutaminase Inhibitors Showed Improved Cellular Uptake and Antitumor Activity.EBI Zhejiang University
31199640 50 Discovery of a Thiadiazole-Pyridazine-Based Allosteric Glutaminase 1 Inhibitor Series That Demonstrates Oral Bioavailability and Activity in Tumor Xenograft Models.EBI AstraZeneca
31324513 2 Design and synthesis of biotinylated Hexylselen as a probe to identify KGA allosteric inhibitors by a convenient biomolecular interaction assay.EBI Zhejiang University
31603674 48 Development and Characterization of a Fluorescent Probe for GLS1 and the Application for High-Throughput Screening of Allosteric Inhibitors.EBI China Pharmaceutical University
30522056 38 Discovery and development of small molecule modulators targeting glutamine metabolism.EBI China Pharmaceutical University
29969024 75 Recent Progress in the Discovery of Allosteric Inhibitors of Kidney-Type Glutaminase.EBI TBA
7664823 5 Modulation of [35S]TBPS binding by ligands with preferential affinity for benzodiazepine BZ1 sites in the cerebral cortex of newborn and adult rats.BDB University of Cagliari
20486938 16 Carbonic anhydrase inhibitors: Inhibition of human erythrocyte isozymes I and II with a series of phenolic acids.BDB Ataturk University
1704434 16 Pharmacologic comparison of selected agonists for the M1 muscarinic receptor in transfected murine fibroblast cells (B82).BDB University of Arizona
18394907 23 Effects of modifications of the linker in a series of phenylpropanoic acid derivatives: Synthesis, evaluation as PPARalpha/gamma dual agonists, and X-ray crystallographic studies.BDB Pfizer Inc
15837304 132 Dipeptidyl peptidase IV inhibitors derived from beta-aminoacylpiperidines bearing a fused thiazole, oxazole, isoxazole, or pyrazole.BDB Merck Research Laboratories
9865942 11 Structural analysis of inhibitor binding to human carbonic anhydrase II.BDB University of Pennsylvania