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19 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
27326325 44 GSK6853, a Chemical Probe for Inhibition of the BRPF1 Bromodomain.EBI GlaxoSmithKline
26572217 60 Disrupting Acetyl-Lysine Recognition: Progress in the Development of Bromodomain Inhibitors.EBI Genentech
26061247 71 Structure-Guided Design of IACS-9571, a Selective High-Affinity Dual TRIM24-BRPF1 Bromodomain Inhibitor.EBI The University of Texas M.D. Anderson Cancer Center
25974391 78 Discovery of a Chemical Tool Inhibitor Targeting the Bromodomains of TRIM24 and BRPF.EBI University of Oxford
26230603 176 Structure-Based Optimization of Naphthyridones into Potent ATAD2 Bromodomain Inhibitors.EBI GlaxoSmithKline
25408830 43 1,3-Dimethyl Benzimidazolones Are Potent, Selective Inhibitors of the BRPF1 Bromodomain.EBI GlaxoSmithKline
25249180 146 The discovery of I-BET726 (GSK1324726A), a potent tetrahydroquinoline ApoA1 up-regulator and selective BET bromodomain inhibitor.EBI GlaxoSmithKline
29656650 151 Discovery of Tetrahydroquinoxalines as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the Second Bromodomain.EBI University of Strathclyde
29169673 115 Design and synthesis of a biaryl series as inhibitors for the bromodomains of CBP/P300.EBI WuXi AppTec Co., Ltd.
28463487 185 Structure-Based Discovery of 4-(6-Methoxy-2-methyl-4-(quinolin-4-yl)-9H-pyrimido[4,5-b]indol-7-yl)-3,5-dimethylisoxazole (CD161) as a Potent and Orally Bioavailable BET Bromodomain Inhibitor.EBI University of Michigan
30015487 96 Structure-Based Discovery of CF53 as a Potent and Orally Bioavailable Bromodomain and Extra-Terminal (BET) Bromodomain Inhibitor.EBI TBA
28068087 80 Design of a Biased Potent Small Molecule Inhibitor of the Bromodomain and PHD Finger-Containing (BRPF) Proteins Suitable for Cellular and in Vivo Studies.EBI University College London
27935314 4 A Versatile Method to Determine the Cellular Bioavailability of Small-Molecule Inhibitors.EBI H. Lee Moffitt Cancer Center and Research Institute
28402630 187 Benzoisoquinolinediones as Potent and Selective Inhibitors of BRPF2 and TAF1/TAF1L Bromodomains.EBI Bayer AG
28268136 130 Methylpyrrole inhibitors of BET bromodomains.EBI AbbVie Inc
28714688 105 Design of a Chemical Probe for the Bromodomain and Plant Homeodomain Finger-Containing (BRPF) Family of Proteins.EBI University College London
12044152 4 DNA gyrase interaction with coumarin-based inhibitors: the role of the hydroxybenzoate isopentenyl moiety and the 5'-methyl group of the noviose.BDB UMR CNRS 6032