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35 articles for thisTarget

The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
24972724 16 Influence of azide incorporation on binding affinity by small papain inhibitors.EBI Radboud University Nijmegen
24077527 11 Squaric acid/4-aminoquinoline conjugates: novel potent antiplasmodial agents.EBI University of Lisbon. Av. Prof. Gama Pinto
23834438 10 Design, synthesis, and optimization of novel epoxide incorporating peptidomimetics as selective calpain inhibitors.EBI University of Illinois College of Pharmacy
23611656 9 Inhibition of rhodesain as a novel therapeutic modality for human African trypanosomiasis.EBI Universit£ degli Studi di Milano
9804696 2 Use of papain as a model for the structure-based design of cathepsin K inhibitors: crystal structures of two papain-inhibitor complexes demonstrate binding to S'-subsites.EBI SmithKline Beecham Pharmaceuticals
22884354 36 Tanshinones as selective and slow-binding inhibitors for SARS-CoV cysteine proteases.EBI Korea Research Institute of Bioscience and Biotechnology
19715320 87 Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation.EBI University of Florida
18995931 16 Natural polyprenylated benzophenones inhibiting cysteine and serine proteases.EBI Federal University of Alfenas
10669559 180 Protease inhibitors: current status and future prospects.EBI University of Queensland
9873373 20 Peptidyl beta-homo-aspartals: specific inhibitors of interleukin-1 beta converting enzyme and its homologues (caspases).EBI Institute for Drug Research
22019466 13 Design, synthesis and biological evaluation of peptidyl-vinylaminophosphonates as novel cysteine protease inhibitors.EBI National Chemical Laboratory (CSIR-NCL)
22071522 6 Aza vinyl sulfones: synthesis and evaluation as antiplasmodial agents.EBI University of Lisbon
21923104 12 HLE-inhibitory alkaloids with a polyketide skeleton from the marine-derived fungus Coniothyrium cereale.EBI University of Bonn
19913414 7 Antimalarial activity of azadipeptide nitriles.EBI University of Queensland
19908842 84 Identification and optimization of inhibitors of Trypanosomal cysteine proteases: cruzain, rhodesain, and TbCatB.EBI National Human Genome Research Institute
 4 Design of a new selective cysteine protease inactivator and its mechanistic implicationsEBI TBA
18789705 6 Peptidyl epoxides extended in the P' direction as cysteine protease inhibitors: effect on affinity and mechanism of inhibition.EBI Bar Ilan University
16759084 12 Isatin compounds as noncovalent SARS coronavirus 3C-like protease inhibitors.EBI Peking University
12213061 23 Azapeptides structurally based upon inhibitory sites of cystatins as potent and selective inhibitors of cysteine proteases.EBI University of Gda£?sk
11720861 24 Discovery, total synthesis, HRV 3C-protease inhibitory activity, and structure-activity relationships of 2-methoxystypandrone and its analogues.EBI Merck Research Laboratories
11141092 85 Novel, nonpeptidic cyanamides as potent and reversible inhibitors of human cathepsins K and L.EBI Merck Frosst Centre for Therapeutic Research
11128643 4 (S)-Thiirancarboxylic acid as a reactive building block for a new class of cysteine protease inhibitors.EBI University of Würzburg
10508448 11 Combinatorial library of serine and cysteine protease inhibitors that interact with both the S and S' binding sites.EBI Brown University
8765519 6 Mechanistic studies on the inactivation of papain by epoxysuccinyl inhibitors.EBI University of Wisconsin
8230139 164 Peptide alpha-keto ester, alpha-keto amide, and alpha-keto acid inhibitors of calpains and other cysteine proteases.EBI School of Chemistry and Biochemistry
7932558 30 Nonpeptidic inhibitors of human leukocyte elastase. 2. Design, synthesis, and in vitro activity of a series of 3-amino-6-arylopyridin-2-one trifluoromethyl ketones.EBI ZENECA Pharmaceuticals Group
7562931 41 Peptidyl alpha-ketoheterocyclic inhibitors of human neutrophil elastase. 3. In vitro and in vivo potency of a series of peptidyl alpha-ketobenzoxazoles.EBI ZENECA Pharmaceuticals
6547487 3 Vinylogous amino acid esters: a new class of inactivators for thiol proteases.EBI TBA
3941405 15 Carboxyl-modified amino acids and peptides as protease inhibitors.EBI TBA
2724298 11 Acid-sensitive latent inhibitors for proteolytic enzymes: synthesis and characterization.EBI Amherst College
15734651 135 A neoceptor approach to unraveling microscopic interactions between the human A2A adenosine receptor and its agonists.BDB National Institutes of Health