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36 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
27287367 36 Evaluation of bisbenzamidines as inhibitors for matriptase-2.EBI University of Bonn
26114810 8 Synthesis of 3,4-diaminobenzoyl derivatives as factor Xa inhibitors.EBI Southeast University
25650311 76 Synthesis and pharmacological characterization of 2-aminobenzaldehyde oxime analogs as dual inhibitors of neutrophil elastase and proteinase 3.EBI Chang Gung University
25268757 16 How aß-D-glucoside side chain enhances binding affinity to thrombin of inhibitors bearing 2-chlorothiophene as P1 moiety: crystallography, fragment deconstruction study, and evaluation of antithrombotic properties.EBI Consiglio Nazionale delle Ricerche
1271404 55 Novel bis(benzamidino) compounds with an aromatic central link. Inhibitors of thrombin, pancreatic kallikrein, trypsin, and complement.EBI TBA
671460 122 Diarylamidine derivatives with one or both of the aryl moieties consisting of an indole or indole-like ring. Inhibitors of arginine-specific esteroproteases.EBI TBA
660589 3 Inactivation of trypsin-like proteases by sulfonylation. Variation of positively charged group and inhibitor length.EBI TBA
24102612 105 Synthesis and biological evaluation of direct thrombin inhibitors bearing 4-(piperidin-1-yl)pyridine at the P1 position with potent anticoagulant activity.EBI University of Bari "Aldo Moro"
7401110 109 Thrombin inhibitors. 2. Amide derivatives of N alpha-substituted L-arginine.EBI TBA
7401109 32 Thrombin inhibitors. 1. Ester derivatives of N alpha-(arylsulfonyl)-L-arginine.EBI TBA
7452681 81 Thrombin inhibitors. 3. Carboxyl-containing amide derivatives of N alpha-substituted L-arginine.EBI TBA
22950366 6 Thrombin inhibitors from the freshwater cyanobacterium Anabaena compacta.EBI Hokkaido University
20561792 4 Development of tryptase inhibitors derived from thalidomide.EBI The University of Tokyo
12036355 36 Simple, intuitive calculations of free energy of binding for protein-ligand complexes. 1. Models without explicit constrained water.EBI University of Parma
11297451 21 Estimation of binding affinities for selective thrombin inhibitors via Monte Carlo simulations.EBI Yale University
10956211 14 GRID/CPCA: a new computational tool to design selective ligands.EBI Boehringer Ingelheim Pharma KG
10579821 51 Design and synthesis of thrombin inhibitors: analogues of MD-805 with reduced stereogenicity and improved potency.EBI Novartis Horsham Research Centre
9301673 234 Synthesis and structure-activity relationships of potent thrombin inhibitors: piperazides of 3-amidinophenylalanine.EBI Klinikum der Friedrich-Schiller-Universit£t Jena
8478905 53 Inhibition studies of some serine and thiol proteinases by new leupeptin analogues.EBI University of Arkansas
3625715 18 Anticoagulant peptides: nature of the interaction of the C-terminal region of hirudin with a noncatalytic binding site on thrombin.EBI TBA
19193009 25 Fluorinated benzyloxyphenyl piperidine-4-carboxamides with dual function against thrombosis: inhibitors of factor Xa and platelet aggregation.EBI University of Bari
 19 Rational design of selective thrombin inhibitorsEBI TBA
 61 (N-acyl-N-alkyl)glycyl borolysine analogs: A new class of potent thrombin inhibitorsEBI TBA
 13 Characterization of LY806303 as a potent and selective inhibitor of thrombinEBI TBA
9834152 29 Effects of tannins from Geum japonicum on the catalytic activity of thrombin and factor Xa of blood coagulation cascade.EBI National University of Singapore
11549459 5 Synthesis and evaluation of the sunflower derived trypsin inhibitor as a potent inhibitor of the type II transmembrane serine protease, matriptase.EBI National Cancer Institute
9876114 111 Structural and functional analyses of benzamidine-based inhibitors in complex with trypsin: implications for the inhibition of factor Xa, tPA, and urokinase.EBI Institut für Biochemie
9871573 15 Discovery of LB30057, a benzamidrazone-based selective oral thrombin inhibitor.EBI Biotech Research Institute
9784099 84 Design of benzamidine-type inhibitors of factor Xa.EBI Institut für Biochemie
7473571 90 Structure-activity study of tripeptide thrombin inhibitors using alpha-alkyl amino acids and other conformationally constrained amino acid substitutions.EBI Lilly Research Laboratories
6219223 94 Aromatic amidines: comparison of their ability to block respiratory syncytial virus induced cell fusion and to inhibit plasmin, urokinase, thrombin, and trypsin.EBI TBA