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18 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
27287367 36 Evaluation of bisbenzamidines as inhibitors for matriptase-2.EBI University of Bonn
26421993 44 Structure-guided discovery of 2-aryl/pyridin-2-yl-1H-indole derivatives as potent and selective hepsin inhibitors.EBI Aurigene Discovery Technologies Limited
24794746 168 Structure-guided discovery of 1,3,5 tri-substituted benzenes as potent and selective matriptase inhibitors exhibiting in vivo antitumor efficacy.EBI Aurigene Discovery Technologies Limited
20503967 138 Factor Xa inhibitors: next-generation antithrombotic agents.EBI Bristol-Myers Squibb Company
10956211 14 GRID/CPCA: a new computational tool to design selective ligands.EBI Boehringer Ingelheim Pharma KG
9301673 234 Synthesis and structure-activity relationships of potent thrombin inhibitors: piperazides of 3-amidinophenylalanine.EBI Klinikum der Friedrich-Schiller-Universit£t Jena
10498204 25 Aminoisoquinolines: design and synthesis of an orally active benzamidine isostere for the inhibition of factor XA.EBI Rh£ne-Poulenc Rorer
19805567 3 Long-lasting enfuvirtide carrier pentasaccharide conjugates with potent anti-human immunodeficiency virus type 1 activity.EBI Endotis Pharma
 32 Bisbenzamidine isoxazoline derivatives as factor Xa inhibitorsEBI TBA
 13 Characterization of LY806303 as a potent and selective inhibitor of thrombinEBI TBA
16970403 74 Diphenyl phosphonate inhibitors for the urokinase-type plasminogen activator: optimization of the P4 position.EBI University of Antwerp
12036353 38 Design of selective thrombin inhibitors based on the (R)-Phe-Pro-Arg sequence.EBI Pfizer Global Research and Development
10636232 58 Design, synthesis and structure-activity relationship of a series of arginine aldehyde factor Xa inhibitors. Part 1: structures based on the (D)-Arg-Gly-Arg tripeptide sequence.EBI COR Therapeutics, Inc.
10560742 85 3-Amidinophenylalanine-based inhibitors of urokinase.EBI Universität Jena
9876114 111 Structural and functional analyses of benzamidine-based inhibitors in complex with trypsin: implications for the inhibition of factor Xa, tPA, and urokinase.EBI Institut für Biochemie
9784099 84 Design of benzamidine-type inhibitors of factor Xa.EBI Institut für Biochemie
7473571 90 Structure-activity study of tripeptide thrombin inhibitors using alpha-alkyl amino acids and other conformationally constrained amino acid substitutions.EBI Lilly Research Laboratories