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31 articles for thisTarget

The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
28603989 53 a-Conotoxin [S9A]TxID Potently Discriminates betweena34 anda6/a34 Nicotinic Acetylcholine Receptors.EBI Hainan University
28337332 41 BMS-933043, a Selectivea7 nAChR Partial Agonist for the Treatment of Cognitive Deficits Associated with Schizophrenia.EBI Bristol-Myers Squibb
27958732 93 Design and Synthesis of a New Series of 4-Heteroarylamino-1'-azaspiro[oxazole-5,3'-bicyclo[2.2.2]octanes asa7 Nicotinic Receptor Agonists. 1. Development of Pharmacophore and Early Structure-Activity Relationship.EBI Bristol-Myers Squibb
27639361 88 Synthesis and biological evaluation of novel hybrids of highly potent and selectivea42-Nicotinic acetylcholine receptor (nAChR) partial agonists.EBI University of Illinois at Chicago
24844195 21 Synthesis and pharmacological characterization of new neuronal nicotinic acetylcholine receptor ligands derived from Sazetidine-A.EBI Georgetown University Medical Center
24187998 96 Design, synthesis, and biological evaluation of Erythrina alkaloid analogues as neuronal nicotinic acetylcholine receptor antagonists.EBI University of Copenhagen
24649848 47 Discovery of a potent and selectivea34 nicotinic acetylcholine receptor antagonist from ana-conotoxin synthetic combinatorial library.EBI Torrey Pines Institute for Molecular Studies
15050615 36 Synthesis and pharmacological characterization of bivalent ligands of epibatidine at neuronal nicotinic acetylcholine receptors.EBI University of Illinois at Chicago
24428686 6 Synthesis, nicotinic acetylcholine receptor binding, and antinociceptive properties of 2'-fluoro-3'-(substituted pyridinyl)-7-deschloroepibatidine analogues.EBI Research Triangle Institute
24274400 28 Scaffold ranking and positional scanning utilized in the discovery of nAChR-selective compounds suitable for optimization studies.EBI Torrey Pines Institute for Molecular Studies
24200193 32 Characterization of a novela-conotoxin TxID from Conus textile that potently blocks rata34 nicotinic acetylcholine receptors.EBI Hainan University
24047231 52 Design, synthesis and discovery of picomolar selective α4β2 nicotinic acetylcholine receptor ligands.EBI Georgetown University
15686946 36 Halogenated and isosteric cytisine derivatives with increased affinity and functional activity at nicotinic acetylcholine receptors.EBI National Institute of Diabetes and Digestive and Kidney Diseases
22410083 17 Consequences of linker length alteration of thea7 nicotinic acetylcholine receptor (nAChR) agonist, SEN12333.EBI The University of Sydney
18989912 95 Novel acetylcholine and carbamoylcholine analogues: development of a functionally selective alpha4beta2 nicotinic acetylcholine receptor agonist.EBI University of Copenhagen
18605717 41 Discovery of (-)-7-methyl-2-exo-[3'-(6-[18F]fluoropyridin-2-yl)-5'-pyridinyl]-7-azabicyclo[2.2.1]heptane, a radiolabeled antagonist for cerebral nicotinic acetylcholine receptor (alpha4beta2-nAChR) with optimal positron emission tomography imaging properties.EBI The Johns Hopkins UniVersity School of Medicine
15050613 50 Pharmacology of the agonist binding sites of rat neuronal nicotinic receptor subtypes expressed in HEK 293 cells.EBI Georgetown University School of Medicine
11354387 20 Neuronal nicotinic acetylcholine receptor binding affinities of boron-containing nicotine analogues.EBI University of Kentucky
20979364 40 Novela3ß4 nicotinic acetylcholine receptor-selective ligands. Discovery, structure-activity studies, and pharmacological evaluation.EBI SRI International
19481945 55 Synthesis and biological evaluation of novel carbon-11 labeled pyridyl ethers: candidate ligands for in vivo imaging of alpha4beta2 nicotinic acetylcholine receptors (alpha4beta2-nAChRs) in the brain with positron emission tomography.EBI The Johns Hopkins University School of Medicine
17067175 3 Isolation, structure elucidation, and biological evaluation of 15-amido-3-demethoxy-2alpha,3alpha-methylenedioxyerythroculine, a new alkaloid from Hyperbaena valida.EBI GlaxoSmithKline Pharmaceuticals
16005216 20 The characterization of a novel rigid nicotine analog with alpha7-selective nAChR agonist activity and modulation of agonist properties by boron inclusion.EBI University of Florida
15771418 38 Novel pyridyl ring C5 substituted analogues of epibatidine and 3-(1-methyl-2(S)-pyrrolidinylmethoxy)pyridine (A-84543) as highly selective agents for neuronal nicotinic acetylcholine receptors containing beta2 subunits.EBI University of Illinois at Chicago
15050621 100 Epibatidine structure-activity relationships.EBI Research Triangle Institute
14971903 17 Chemical and functional identification and characterization of novel sulfated alpha-conotoxins from the cone snail Conus anemone.EBI The University of Queensland
29178785 61 Highly Selective and Potent?4?2 nAChR Antagonist Inhibits Nicotine Self-Administration and Reinstatement in Rats.EBI Torrey Pines Institute for Molecular Studies