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24 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
6292417 10 Hydroxy- and amino-substituted piperidinecarboxylic acids as gamma-aminobutyric acid agonists and uptake inhibitors.EBI TBA
27654218 56 Synthesis and biological evaluation of a series of N-alkylated imidazole alkanoic acids as mGAT3 selective GABA uptake inhibitors.EBI Ludwig-Maximilians-Universit£t M£nchen
27039250 58 Synthesis of 4-substituted nipecotic acid derivatives and their evaluation as potential GABA uptake inhibitors.EBI Ludwig-Maximilians-Universit£t M£nchen
26706177 136 Straightforward and effective synthesis of┐-aminobutyric acid transporter subtype 2-selective acyl-substituted azaspiro[4.5]decanes.EBI Universit£ catholique de Louvain
25679268 9 A binding mode hypothesis of tiagabine confirms liothyronine effect on┐-aminobutyric acid transporter 1 (GAT1).EBI University of Vienna
25882526 496 Structure activity relationship of selective GABA uptake inhibitors.EBI University of Copenhagen
25698617 61 Design, synthesis and SAR studies of GABA uptake inhibitors derived from 2-substituted pyrrolidine-2-yl-acetic acids.EBI Ludwig-Maximilians-Universit£t M£nchen
25025595 30 First photoswitchable neurotransmitter transporter inhibitor: light-induced control of┐-aminobutyric acid transporter 1 (GAT1) activity in mouse brain.EBI Ludwig-Maximilians-Universit£t M£nchen
24973660 150 Synthesis, biological evaluation and structure-activity relationship of new GABA uptake inhibitors, derivatives of 4-aminobutanamides.EBI Jagiellonian University Medical College
23398473 85 Selective mGAT2 (BGT-1) GABA uptake inhibitors: design, synthesis, and pharmacological characterization.EBI University of Copenhagen
23336362 10 Focused pseudostatic hydrazone libraries screened by mass spectrometry binding assay: optimizing affinities toward¿-aminobutyric acid transporter 1.EBI Ludwig Maximilians University at Munich
21940173 32 Aminomethyltetrazoles as potential inhibitors of the¿-aminobutyric acid transporters mGAT1-mGAT4: synthesis and biological evaluation.EBI Ludwig-Maximilians-University Munich
17517506 14 Synthesis and biological evaluation of (R)-N-(diarylmethylthio/sulfinyl)ethyl/propyl-piperidine-3-carboxylic acid hydrochlorides as novel GABA uptake inhibitors.EBI Zhengzhou University
16821765 29 Development of peptidic dopamine transporter inhibitors via aromatic modification-mediated conformational restriction.EBI Chinese Academy of Sciences
15509161 90 Novel secoergoline derivatives inhibit both GABA and glutamate uptake in rat brain homogenates: synthesis, in vitro pharmacology, and modeling.EBI Budapest University of Technology and Economics
10543872 31 Synthesis of novel GABA uptake inhibitors. 4. Bioisosteric transformation and successive optimization of known GABA uptake inhibitors leading to a series of potent anticonvulsant drug candidates.EBI Novo Nordisk A/S
10479278 70 Synthesis of novel GABA uptake inhibitors. 3. Diaryloxime and diarylvinyl ether derivatives of nipecotic acid and guvacine as anticonvulsant agents.EBI Novo Nordisk A/S
6304315 8 4,5,6,7-Tetrahydroisothiazolo[5,4-c]pyridin-3-ol and related analogues of THIP. Synthesis and biological activity.EBI TBA
21353350 61 Development of imidazole alkanoic acids as mGAT3 selective GABA uptake inhibitors.EBI Ludwig-Maximilians-University Munich
19703775 24 Synthesis and biological evaluation of 4-fluoroproline and 4-fluoropyrrolidine-2-acetic acid derivatives as new GABA uptake inhibitors.EBI Institute of Microbiology
 20 On the bioactive conformation of the gaba uptake inhibitor SK&F 89976-AEBI TBA
18395300 1 Synthesis and biological evaluation of aminomethylphenol derivatives as inhibitors of the murine GABA transporters mGAT1-mGAT4.EBI Ludwig-Maximilians-Universität München
8057281 100 Design, synthesis and evaluation of substituted triarylnipecotic acid derivatives as GABA uptake inhibitors: identification of a ligand with moderate affinity and selectivity for the cloned human GABA transporter GAT-3.EBI Synaptic Pharmaceutical Corporation
2999396 12 GABA agonists. Resolution, absolute stereochemistry, and enantioselectivity of (S)-(+)- and (R)-(-)-dihydromuscimol.EBI TBA