BDBM50210259 (4Z,7Z,10Z,13Z,16Z,19Z)-docosa-4,7,10,13,16,19-hexaenoic acid::(4Z,7Z,10Z,13Z,16Z,19Z)-docosa-4,7,10,13,16,19-hexaenoic acid (F4)::CHEMBL367149::DHA::Doconexent::all-cis-docosa-4,7,10,13,16,19-hexaenoic acid
SMILES CC\C=C/C\C=C/C\C=C/C\C=C/C\C=C/C\C=C/CCC(O)=O
InChI Key InChIKey=MBMBGCFOFBJSGT-KUBAVDMBSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 10 hits for monomerid = 50210259
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Okayama University Graduate School Of Medicine
Curated by ChEMBL
Okayama University Graduate School Of Medicine
Curated by ChEMBL
Affinity DataKi: 6.29E+3nMAssay Description:Displacement of CU-6PMN from human RXRalpha LBD incubated for 2 hrs by fluorescence based assayMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Okayama University Graduate School Of Medicine
Curated by ChEMBL
Okayama University Graduate School Of Medicine
Curated by ChEMBL
Affinity DataKi: 6.29E+3nMAssay Description:Displacement of CU-6PMN from human RXRalpha LBD incubated for 2 hrs by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.17E+4nMAssay Description:Agonist activity at GPR40 (unknown origin) by Fluo-4 AM dye based calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at human OXE receptor fused with G-alphai assessed as inhibition of 5-oxo-ETE-induced GTPgammaS binding after 60 mins by liquid s...More data for this Ligand-Target Pair
Affinity DataEC50: 3.60E+4nMAssay Description:Agonist activity at GPR40 expressed in CHO cells after 20 seconds by aequorin bioluminescence assay in presence of 0.1 % human serumMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of bovine COX1-mediated prostaglandin biosynthesis using [1-14C]arachidonic acidMore data for this Ligand-Target Pair
Affinity DataIC50: 9.80E+3nMAssay Description:Inhibition of sheep COX2-mediated prostaglandin biosynthesis using [1-14C]arachidonic acidMore data for this Ligand-Target Pair
Affinity DataIC50: 6.76E+3nMpH: 7.5 T: 2°CAssay Description:All assays were performed at 100 µL total volume in triplicate and monitored for 60 minutes at room temperature in a 96-well plate format in HEPES Bu...More data for this Ligand-Target Pair
Affinity DataIC50: 3.32E+4nMAssay Description:Inhibition of aromatase in human placental microsomes by radiometric methodMore data for this Ligand-Target Pair