BDBM50221813 CHEMBL394602::HO-LVA
SMILES [#6]-[#7](-[#6@H](-[#6]-c1ccc(-[#8])cc1)-[#6](=O)-[#7]-[#6@@H](-[#6]-c1ccccc1)-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6](-[#7])=O)-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6](-[#7])=O)-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7])-[#6](=O)-[#7]-1-[#6]-[#6]-[#6@@H](-[#6]-1)-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7])-[#6](-[#7])=O)-[#6](=O)-[#6]-c1ccc(-[#8])cc1
InChI Key InChIKey=QSWYUUWOWAFPRH-PDQNOIBYSA-N
Data 5 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50221813
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.0320nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in CHO cells by polarisation binding assay using 384-well plate membranesMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.0360nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in CHO cells by polarisation binding assay using 96-well plate membranesMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.210nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in COS7 cells by HTRF-FRET assay using 384-well plate membranesMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.210nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in COS7 cells by HTRF-FRET assay using 96-well plate membranesMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.280nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in COS7 cells by HTRF-FRET assay using 96-well plate cellsMore data for this Ligand-Target Pair