BDBM10127 tert-butyl N-(2-{[9-fluoro-3-oxo-5-(1H-pyrrol-2-yl)-2-azatricyclo[6.3.1.0^{4,12}]dodeca-1(11),4,6,8(12),9-pentaen-7-yl]amino}ethyl)carbamate::trisubstituted naphthostyril analogue 7g
SMILES CC(C)(C)OC(=O)NCCNc1cc(-c2ccc[nH]2)c2C(=O)Nc3ccc(F)c1c23
InChI Key InChIKey=HUUYQUKEWGQKGJ-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 10127
Affinity DataIC50: 5.50E+3nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed using a recombinant human cyclin E-CDK2 complex. The enzyme was assayed with substrate in the presence of 1uM ATP/[gamma...More data for this Ligand-Target Pair