BDBM112592 US8618103, I-88
SMILES CSc1ncc(c(N[C@H]2CCCN(C2)C(=O)CC#N)n1)-c1cnc2[nH]ccc2n1
InChI Key InChIKey=VCPJACUOLDMQIU-LBPRGKRZSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 112592
Affinity DataKi: 0.422nM IC50: 0.844nMpH: 7.2Assay Description:The kinase activity of all three JAK kinases is measured using a radioactive, end-point assay and with trace amounts of 33P-ATP. More data for this Ligand-Target Pair
Affinity DataIC50: 0.223nMpH: 7.2Assay Description:The kinase activity of all three JAK kinases is measured using a radioactive, end-point assay and with trace amounts of 33P-ATP. More data for this Ligand-Target Pair