BDBM120222 US8691753, 71
SMILES OC(=O)CC[C@H](NC(=O)CCc1ccc(cc1)-c1ccc(cc1)-c1ccccc1)C(=O)Nc1cccc(CC(O)=O)c1
InChI Key InChIKey=OUZMHHWAGJCAFA-PMERELPUSA-N
Data 8 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 120222
TargetMacrophage metalloelastase(Homo sapiens (Human))
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Affinity DataKi: 1.05nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
TargetStromelysin-2(Homo sapiens (Human))
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Affinity DataKi: 7.70nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
TargetCollagenase 3(Homo sapiens (Human))
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Affinity DataKi: 10.2nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Affinity DataKi: 18.1nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
TargetStromelysin-1(Homo sapiens (Human))
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Affinity DataKi: 34nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
TargetNeutrophil collagenase(Homo sapiens (Human))
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Affinity DataKi: 99nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Affinity DataKi: 645nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-14 [1-20,P8S](Homo sapiens (Human))
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Commissariat A L'Energie Atomique Et Aux Energies Alternatives
US Patent
Affinity DataKi: 696nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair