BDBM121143 US8722896, (+/-)-2-Methyl-3-((2- hydroxybenzyl)methylamino)-N- (9-chloro-3,4-dihydro-2H-1,5- benzodioxepin-7-ylmethyl)-N- isobutylpropanamide
SMILES CC(C)CN(Cc1cc(Cl)c2OCCCOc2c1)C(=O)C(C)CNCc1cccc(O)c1
InChI Key InChIKey=HCMJCMYVOXIEMD-UHFFFAOYSA-N
Data 4 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 121143
TargetProkineticin receptor 2(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California
US Patent
The Regents Of The University Of California
US Patent
Affinity DataKi: 1.62nM ΔG°: -12.5kcal/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
TargetProkineticin receptor 2(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California
US Patent
The Regents Of The University Of California
US Patent
Affinity DataKi: 1.77nM ΔG°: -12.4kcal/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California
US Patent
The Regents Of The University Of California
US Patent
Affinity DataKi: 7.80nM ΔG°: -11.5kcal/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents Of The University Of California
US Patent
The Regents Of The University Of California
US Patent
Affinity DataKi: 23.5nM ΔG°: -10.8kcal/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair