BDBM122706 US8735386, I-176

SMILES COc1ccc(cc1)-c1c-2c(CCc3cnc(Nc4cnn(c4)C4CCN(CC4)C(C)=O)nc-23)nn1C

InChI Key InChIKey=TVPNAVAKVYZWEN-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 122706   

TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM122706(US8735386, I-176)
Affinity DataIC50:  0.400nMpH: 7.4Assay Description:The kinase activity is measured by DELFIA assay (dissociation-enhanced lanthanide fluorescence immunoassay, Perkin Elmer). The cytoplasmic kinase dom...More data for this Ligand-Target Pair
In DepthDetails US Patent