BDBM129567 US8802673, 209
SMILES Fc1cnc(Nc2ccc(C3CNCCO3)c(F)c2)nc1OCC(F)(F)F
InChI Key InChIKey=ALNGRRMJEIRAFV-UHFFFAOYSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 129567
Affinity DataKi: 2.5nM ΔG°: -12.2kcal/molepH: 7.4 T: 37°CAssay Description:HEK-293 cells stably expressing mouse TAAR1 were maintained at 37 C. and 5% CO2 in DMEM high glucose medium, containing fetal calf serum (10%, heat i...More data for this Ligand-Target Pair
Affinity DataKi: 3.20nM ΔG°: -12.0kcal/molepH: 7.4 T: 37°CAssay Description:HEK-293 cells stably expressing rat TAAR1 were maintained at 37 C. and 5% CO2 in DMEM high glucose medium, containing fetal calf serum (10%, heat ina...More data for this Ligand-Target Pair