BDBM144278 US8969333, YW4-15
SMILES CN(C)c1ccc2cc(ccc2c1)C(=O)N[C@@H](CCCNC(=N)CCl)C(=O)NCc1ccc(NC(=O)CCCNC(=O)CCCCC2SCC3NC(=O)NC23)cc1
InChI Key InChIKey=PZYFZMCZZMDILQ-RQWDCHKRSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 144278
TargetProtein-arginine deiminase type-6(Homo sapiens (Human))
The Penn State Research Foundation
US Patent
The Penn State Research Foundation
US Patent
Affinity DataIC50: 3.50E+3nMT: 2°CAssay Description:The inhibition efficacy of PAD4 inhibitors were determined by colorimetric measurement of citrulline generated by PAD4 catalyzed citrullination of BA...More data for this Ligand-Target Pair