BDBM148134 US8962609, DMX-75
SMILES Cn1cc(Nc2nccc(n2)-c2ccc(N3CCC(CC3)C(N)=O)c(c2)C#N)cn1
InChI Key InChIKey=DQGNBSROXUZAHD-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 148134
Affinity DataIC50: <300nMpH: 7.5Assay Description:Inhibitions studies were performed using a time-resolved fluorescence-based Lanthascreen assay. Phosphorylation of a fluorescein-labelled substrate p...More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Domainex
US Patent
Domainex
US Patent
Affinity DataIC50: <30nMpH: 7.5Assay Description:Inhibitions studies were performed using a time-resolved fluorescence-based Lanthascreen assay. Phosphorylation of a fluorescein-labelled substrate p...More data for this Ligand-Target Pair