BDBM152807 BDBM152808::US8993568, 2
SMILES C[C@@H](NS(C)(=O)=O)c1ccc(CN2CCO[C@H](C2)c2ccc(F)cc2)cc1
InChI Key InChIKey=JUONYSHFHZDWHI-FOIQADDNSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 152807
Affinity DataIC50: 44nMT: 2°CAssay Description:The in vitro inhibitory activity of compounds against human MOGAT-2 is evaluated in this assay. MOGAT-2 transfers an oleoyl group to monooleoyl-glyce...More data for this Ligand-Target Pair
TargetAlpha-1,6-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 274nMAssay Description:Inhibition of recombinant human MGAT2 expressed in sf9 cells using 2-monooleoyl glycerol/[14C]-oleoyl CoA as substrate by microscintillation counting...More data for this Ligand-Target Pair
Affinity DataIC50: 274nMT: 2°CAssay Description:The in vitro inhibitory activity of compounds against human MOGAT-2 is evaluated in this assay. MOGAT-2 transfers an oleoyl group to monooleoyl-glyce...More data for this Ligand-Target Pair