BDBM179800 3-((2,6-dichloro-3-fluorophenyl)sulfide)-5-(1-(piperidin-4-yl)-1H-pyrazol-4-yl)-1Hpyrrolo[2,3-b]pyridine (8)
SMILES Fc1ccc(Cl)c(c1Cl)S(=O)c1c[nH]c2ncc(cc12)-c1cnn(c1)C1CCNCC1
InChI Key InChIKey=LEHQHFLLRYUONA-UHFFFAOYSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 179800
TargetIsoform 2 of Hepatocyte growth factor receptor (2)(Homo sapiens (Human))
Tianjin University Of Science And Technology
Tianjin University Of Science And Technology
Affinity DataIC50: 63nMpH: 7.0 T: 2°CAssay Description:The c-Met kinase activity of five target compounds and three positive compounds were evaluated using standard Z-LYTE Assays (fluorescence resonance e...More data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor [L1196M](Homo sapiens (Human))
Tianjin University Of Science And Technology
Tianjin University Of Science And Technology
Affinity DataIC50: 725nMpH: 7.5 T: 2°CAssay Description:The ALK kinase activity of five target compounds and three positive compounds were evaluated using standard homogeneous time-resolved fluorescence (H...More data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor [C1156Y](Homo sapiens (Human))
Tianjin University Of Science And Technology
Tianjin University Of Science And Technology
Affinity DataIC50: 1.31E+3nMpH: 7.5 T: 2°CAssay Description:The ALK kinase activity of five target compounds and three positive compounds were evaluated using standard homogeneous time-resolved fluorescence (H...More data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Tianjin University Of Science And Technology
Tianjin University Of Science And Technology
Affinity DataIC50: 214nMpH: 7.5 T: 2°CAssay Description:The ALK kinase activity of five target compounds and three positive compounds were evaluated using standard homogeneous time-resolved fluorescence (H...More data for this Ligand-Target Pair