BDBM183842 US9150526, 95::US9199947, 104
SMILES Cc1cnc(s1)C(CC(O)=O)c1cc(Cl)cc(c1)-c1ccccc1OC(F)(F)F
InChI Key InChIKey=ZAYXQLJKKJFTDJ-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 183842
Affinity DataIC50: 221nMpH: 5.5 T: 2°CAssay Description:The activated cathepsin A was diluted in assay buffer (25 mM MES, pH 5.5, containing 5 mM DTT) and mixed with the test compound (dissolved in assay b...More data for this Ligand-Target Pair
Affinity DataIC50: 221nMpH: 6.0 T: 2°CAssay Description:Recombinant human cathepsin A (residues 29-480, with a C-terminal 10-His tag; R&D Systems, #1049-SE) was proteolytically activated with recombinant h...More data for this Ligand-Target Pair