BDBM185927 US9163008, 16::US9656968, Compound 16

SMILES CCOC(=O)[C@@H]1Cc2ccccc2N1c1cc(nc(n1)-c1ccc(Oc2ccc(F)cc2)cc1)C(N)=O

InChI Key InChIKey=JZEJXCYTVIVQII-DEOSSOPVSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 185927   

TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM185927(US9163008, 16 | US9656968, Compound 16)
Affinity DataIC50: >2.00E+4nMAssay Description:Assay Buffer: The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM185927(US9163008, 16 | US9656968, Compound 16)
Affinity DataIC50: >2.00E+4nMAssay Description:In vitro assays were performed in a recombinant cell line expressing cDNA encoding the alpha subunit (Nav1.7, SCN9a, PN1, NE) of human Nav1.7 (Access...More data for this Ligand-Target Pair
In DepthDetails US Patent