BDBM203349 US9242981, 84
SMILES Cc1cc(ccn1)-c1n[nH]c2CCN(Cc12)C(=O)NC1CCCN(Cc2c(C)cccc2C)C1
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 203349
Affinity DataIC50: 6.30nMAssay Description:Activated ERK2 activity was also determined in the IMAP assay format using the procedure outlined above. 1 μl of 25× compound was added to 14 ...More data for this Ligand-Target Pair
Affinity DataKd: 0.130nMT: 2°CAssay Description:The SAR (Structure Activity Relationship) for ERK ligands covered by
this invention was interrogated using the TdF (Temperature Dependence
Fluoresc...More data for this Ligand-Target Pair