BDBM20651 4-{[5-(methoxycarbamoyl)-2-methylphenyl]amino}-5-methyl-N-(propan-2-yl)pyrrolo[1,2-a][1,2,4]triazine-6-carboxamide::pyrrolo[2,1-f][1,2,4]triazine analogue, 11d

SMILES CONC(=O)c1ccc(C)c(Nc2ncnn3cc(C(=O)NC(C)C)c(C)c23)c1

InChI Key InChIKey=RELNTJYHSYJKCZ-UHFFFAOYSA-N

Data  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 20651   

TargetMitogen-activated protein kinase 14(Human)
Novartis Pharmaceuticals

LigandPNGBDBM20651(4-{[5-(methoxycarbamoyl)-2-methylphenyl]amino}-5-m...)
Affinity DataIC50:  10nM EC50:  41nMpH: 7.5 T: 22°CAssay Description:The kinase activity was determined by quantitation of the amount of radioactive phosphate transferred to myelin basic protein (MBP) with or without i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed