BDBM209045 US9243038, 20

SMILES NCCCC[C@@H]1NC(=O)\C=C\C(=O)NC(CCCCNC(=O)[C@@H](Cc2ccc(cc2)C(=O)c2ccccc2)NC(=O)[C@H](CC2CCCCC2)NC1=O)C(N)=O

InChI Key InChIKey=BHZABWWULWHRIY-ACWJXPKNSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 209045   

TargetInsulin-degrading enzyme(Mus musculus (Mouse))
President And Fellows Of Harvard College

US Patent
LigandPNGBDBM209045(US9243038, 20)
Affinity DataIC50:  90nMAssay Description:Macrocycles were assayed for IDE inhibition by monitoring cleavage of a substrate peptide containing a fluorophore-quencher pair such that cleavage o...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInsulin-degrading enzyme(Homo sapiens (Human))
President And Fellows Of Harvard College

US Patent
LigandPNGBDBM209045(US9243038, 20)
Affinity DataIC50:  65nMAssay Description:Macrocycles were assayed for IDE inhibition by monitoring cleavage of a substrate peptide containing a fluorophore-quencher pair such that cleavage o...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent