BDBM22545 4-Benzyl-1H-imidazole derivative, 23::4-[(4-bromophenyl)methyl]-1H-imidazole

SMILES Brc1ccc(Cc2cnc[nH]2)cc1

InChI Key InChIKey=WXUFCVQAMIUJMP-UHFFFAOYSA-N

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 22545   

TargetHistamine H3 receptor(Homo sapiens (Human))
Vu University Amsterdam

LigandPNGBDBM22545(4-Benzyl-1H-imidazole derivative, 23 | 4-[(4-bromo...)
Affinity DataKi:  417nM ΔG°:  -8.70kcal/mole EC50:  631nMpH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed