BDBM229716 US9334269, 43

SMILES CNC(=O)c1cccc(Nc2ncnc(n2)N2CCN(CC2)c2cccc(c2)C(F)(F)F)c1

InChI Key InChIKey=HSMTVHSYAURGSR-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 229716   

TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM229716(US9334269, 43)
Affinity DataIC50:  600nMAssay Description:Compounds were tested on human Nav1.7 (hNav1.7) expressed stably in 293 cells, which have no endogenous sodium channels. Two forms of whole-cell patc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent