BDBM230245 US9340500, I-089
SMILES FC(F)(F)c1cccc(Nc2ccc3C(CCCN4CCOCC4)[N](=Cc3c2)c2ccccc2)c1
InChI Key InChIKey=SIIGPTAGWIOOPW-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 230245
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Shionogi
US Patent
Shionogi
US Patent
Affinity DataKi: 3.90E+3nM ΔG°: -7.67kcal/mole IC50: 8.00E+3nMT: 2°CAssay Description:Test Example 1: (1) The TRPV4 inhibitory activity was measured using CHO-K1 cells stably expressing human TRPV4 (hTRPV4/CHO cells). (2) In the day be...More data for this Ligand-Target Pair