BDBM235822 US9364459, J

SMILES COc1cc(cc(OC)c1OC)C1=C(C(=O)NC1=O)c1cn(CCN(C)C)c2ccccc12

InChI Key InChIKey=HXQBEBWEVDQZOZ-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 235822   

TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT Mainz

US Patent
LigandPNGBDBM235822(US9364459, J)
Affinity DataIC50:  1.30E+3nMAssay Description:The effect of test compounds on the activity of the protein kinases GSK-3β, VEGFR-2 and FLT-3 was evaluated based on half maximal inhibitory con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT Mainz

US Patent
LigandPNGBDBM235822(US9364459, J)
Affinity DataIC50:  3.58E+3nMAssay Description:The effect of test compounds on the activity of the protein kinases GSK-3β, VEGFR-2 and FLT-3 was evaluated based on half maximal inhibitory con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT Mainz

US Patent
LigandPNGBDBM235822(US9364459, J)
Affinity DataIC50: >1.00E+3nMAssay Description:The effect of test compounds on the activity of the protein kinases GSK-3β, VEGFR-2 and FLT-3 was evaluated based on half maximal inhibitory con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent