BDBM23908 3-[(2S)-2-(naphthalene-2-sulfonamido)-3-oxo-3-[4-(piperidin-4-yl)piperidin-1-yl]propyl]benzene-1-carboximidamide::3-amidinophenylalanine deriv., 51

SMILES NC(=N)c1cccc(C[C@H](NS(=O)(=O)c2ccc3ccccc3c2)C(=O)N2CCC(CC2)C2CCNCC2)c1

InChI Key InChIKey=QACZHTZZUSYTGR-NDEPHWFRSA-N

Data  5 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 23908   

TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Curacyte Chemistry

LigandPNGBDBM23908(3-[(2S)-2-(naphthalene-2-sulfonamido)-3-oxo-3-[4-(...)
Affinity DataKi:  120nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Curacyte Chemistry

LigandPNGBDBM23908(3-[(2S)-2-(naphthalene-2-sulfonamido)-3-oxo-3-[4-(...)
Affinity DataKi:  210nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Curacyte Chemistry

LigandPNGBDBM23908(3-[(2S)-2-(naphthalene-2-sulfonamido)-3-oxo-3-[4-(...)
Affinity DataKi:  2.20E+3nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Curacyte Chemistry

LigandPNGBDBM23908(3-[(2S)-2-(naphthalene-2-sulfonamido)-3-oxo-3-[4-(...)
Affinity DataKi:  1.20E+4nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Bos taurus)
Curacyte Chemistry

LigandPNGBDBM23908(3-[(2S)-2-(naphthalene-2-sulfonamido)-3-oxo-3-[4-(...)
Affinity DataKi:  2.40E+4nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed