BDBM240690 US9416127, 27
SMILES FC(F)(F)Oc1cccc(c1)-n1cc(nn1)C(=O)Nc1ccc(cc1)[C@H]1CNCCO1
InChI Key InChIKey=SQUVVNMUHMVTFD-GOSISDBHSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 240690
Affinity DataKi: 6.80nM ΔG°: -11.6kcal/molepH: 7.4 T: 2°CAssay Description:HEK-293 cells stably expressing mouse TAAR1 were maintained at 37° C. and 5% CO2 in DMEM high glucose medium, containing fetal calf serum (10%, h...More data for this Ligand-Target Pair
Affinity DataKi: 15.4nMpH: 7.4Assay Description:HEK-293 cells stably expressing rat TAAR1 were maintained at 37° C. and 5% CO2 in DMEM high glucose medium, containing fetal calf serum (10%, heat i...More data for this Ligand-Target Pair