BDBM243282 9-(cyclopropylsulfonyl)-7-((4,4- difluoro-1-piperidinyl)carbonyl)-3- (3,5-dimethyl-4-isoxazolyl)-9H- carbazole-1-carboxamide::US10053454, Example 26::US10196387, Example 26
SMILES Cc1noc(C)c1-c1cc(C(N)=O)c2n(c3cc(ccc3c2c1)C(=O)N1CCC(F)(F)CC1)S(=O)(=O)C1CC1
InChI Key InChIKey=XPLFLWKHNNPZJL-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 243282
Affinity DataIC50: <50nMAssay Description:The binding of compounds to bromodomain BRD4 (44-168), BRD4 (333-460), and BRD4 (1-477 or 44-460) was assessed using a time resolved fluorescent reso...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:The binding of compounds to bromodomain BRD4 (44-168), BRD4 (333-460), and BRD4 (1-477 or 44-460) was assessed using a time resolved fluorescent reso...More data for this Ligand-Target Pair
Affinity DataIC50: <50nMAssay Description:The binding of compounds to bromodomain BRD4 (44-168), BRD4 (333-460), and BRD4 (1-477 or 44-460) was assessed using a time resolved fluorescent reso...More data for this Ligand-Target Pair