BDBM245656 US9428508, 111

SMILES COc1cc(ccc1Nc1nc2NCC(C)(C)c2c(Nc2ccccc2S(=O)(=O)N(C)C)n1)N1CCOCC1

InChI Key InChIKey=AYIHHAZVWSMLSO-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 245656   

TargetProtein-tyrosine kinase 2-beta(Homo sapiens (Human))
Centaurus Biopharma

US Patent
LigandPNGBDBM245656(US9428508, 111)
Affinity DataIC50: <20nMAssay Description:To measure inhibitory activity of FAK/PYK2 inhibitors, compounds were first prepare as a 1 mM stock in 100% DMSO and 3-fold serial dilution was perfo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Centaurus Biopharma

US Patent
LigandPNGBDBM245656(US9428508, 111)
Affinity DataIC50: <20nMAssay Description:To measure inhibitory activity of FAK/PYK2 inhibitors, compounds were first prepare as a 1 mM stock in 100% DMSO and 3-fold serial dilution was perfo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent